SCHEMBL8031501

SCHEMBL8031501

CCCC(C)(CN1CCN(Cc2ccccc2)CC1)Oc1ccc(Cl)cc1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 6/20 0.52
ALDH1A1 P00352 2/20 0.47
DRD4 P21917 1/20 0.47
KDM4E B2RXH2 2/20 0.45
NPC1 O15118 2/20 0.45
TP53 P04637 2/20 0.45
MEN1 O00255 1/20 0.45
KMT2A Q03164 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
TSHR P16473 1/20 0.44
BCHE P06276 1/20 0.42
ACHE P22303 1/20 0.42
PPARG P37231 1/20 0.42
PPARA Q07869 1/20 0.42
RAB9A P51151 1/20 0.42
MC4R P32245 1/20 0.42
LMNA P02545 1/20 0.42
NR1I2 O75469 1/20 0.42
ADORA3 P0DMS8 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8033218 0.92 SIGMAR1 (0.49) SIGMAR1ALDH1A1DRD4KDM4ENPC1
SCHEMBL8029636 0.83 SIGMAR1 (0.59) SIGMAR1ALDH1A1DRD4KDM4ENPC1
SCHEMBL8031456 0.78 PPARG (0.55) SIGMAR1ALDH1A1KDM4EMEN1KMT2A
SCHEMBL8020027 0.77 SIGMAR1 (0.55) SIGMAR1ALDH1A1KDM4ENPC1TP53
SCHEMBL8029641 0.76 ALDH1A1 (0.65) SIGMAR1ALDH1A1KDM4EMEN1KMT2A
SCHEMBL17861674 0.75 PPARA (0.49) ALDH1A1MEN1KMT2ASMN1; SMN2NPSR1
SCHEMBL8020121 0.74 SIGMAR1 (0.56) SIGMAR1ALDH1A1DRD4KDM4ENPC1
SCHEMBL8035713 0.73 MAPK1 (0.57) SIGMAR1ALDH1A1DRD4KDM4ENPC1
SCHEMBL13036529 0.70 SIGMAR1 (0.69) SIGMAR1ALDH1A1DRD4KDM4EKMT2A
SCHEMBL20090429 0.70 SIGMAR1 (0.62) SIGMAR1ALDH1A1DRD4KDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0702010-B1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR (FR) 2000-03-15 EP disclosed
US-5668138-A AFFINITY FOR SIGMA RECEPTORS, CENTRAL NERVOUS SYSTEM DISORDERS ADIR ET COMPAGNIE (FR) 1997-09-16 US disclosed
EP-0702010-A1 Benzopyranderivatives, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1996-03-20 EP disclosed