SCHEMBL8031532

SCHEMBL8031532

C=C(C)NC(=O)/C=C/CN(C)C

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
ITK Q08881 4/20 0.33
EGFR P00533 3/20 0.33
JAK3 P52333 2/20 0.33
BTK Q06187 3/20 0.31
CDK14 O94921 1/20 0.30
CCNY Q8ND76 1/20 0.30
ERBB2 P04626 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16994112 0.79 CHRNB2 (0.33) CHRNB2CHRNB4CHRNA3CHRNA4JAK3
SCHEMBL7928560 0.78 CHRNB2 (0.55) CHRNB2CHRNB4CHRNA3CHRNA4ITK
SCHEMBL27451892 0.78 CHRNB2 (0.55) CHRNB2CHRNB4CHRNA3CHRNA4ITK
SCHEMBL20425354 0.78 CHRNB2 (0.55) CHRNB2CHRNB4CHRNA3CHRNA4ITK
SCHEMBL20206293 0.78 CHRNB2 (0.37) CHRNB2CHRNB4CHRNA3CHRNA4ITK
SCHEMBL23336220 0.77 CHRNB2 (0.36) CHRNB2CHRNB4CHRNA3CHRNA4ITK
SCHEMBL19890610 0.77 CHRNB2 (0.36) CHRNB2CHRNB4CHRNA3CHRNA4ITK
SCHEMBL16665104 0.77 CHRNB2 (0.36) CHRNB2CHRNB4CHRNA3CHRNA4ITK
SCHEMBL12831951 0.76 JAK3 (0.33) CHRNB2CHRNB4CHRNA3CHRNA4ITK
SCHEMBL9070554 0.75 ALDH1A1 (0.37) CHRNB2CHRNB4CHRNA3CHRNA4ITK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010129053-A2 EGFR INHIBITORS AND METHODS OF TREATING DISORDERS DANA FARBER CANCER INSTITUTE (US) 2010-11-11 WO disclosed
WO-2009082701-A1 HCV PROTEASE INHIBITORS AND USES THEREOF AVILA THERAPEUTICS, INC. (US) 2009-07-02 WO disclosed