SCHEMBL8032027

SCHEMBL8032027

Cn1c(Cc2ccc(C#N)cc2)nc2cc(C(=O)C3(C)CCCC3)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACSL1 P33121 2/20 0.43
RORC P51449 2/20 0.42
HDAC6 Q9UBN7 1/20 0.40
IDH1 O75874 7/20 0.40
BCHE P06276 2/20 0.40
CNR2 P34972 2/20 0.40
OPRM1 P35372 1/20 0.40
ITK Q08881 3/20 0.40
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
TYK2 P29597 1/20 0.39
JAK3 P52333 1/20 0.39
AURKA O14965 1/20 0.39
MAP4K4 O95819 1/20 0.39
CHEK2 O96017 1/20 0.39
PRKCG P05129 1/20 0.39
PHKG2 P15735 1/20 0.39
MARK3 P27448 1/20 0.39
FLT3 P36888 1/20 0.39
CSNK1A1 P48729 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8029874 0.99 ACSL1 (0.43) ACSL1RORCHDAC6IDH1BCHE
SCHEMBL7160501 0.86 HDAC6 (0.53) HDAC6F2
Hydrochloric Acid SCHEMBL8026432 0.84 F2 (0.53) F2
Hydrochloric Acid SCHEMBL8016349 0.83 F2 (0.52) F2
SCHEMBL8032232 0.82 ACSL1 (0.42) ACSL1RORCBCHECNR2OPRM1
SCHEMBL8017278 0.81 ITK (0.51) ACSL1CNR2ITKAURKAMAP4K4
SCHEMBL8029791 0.81 RORC (0.45) ACSL1RORCHDAC6IDH1CNR2
SCHEMBL8016519 0.78 F2 (0.55) ACSL1RORCIDH1ITKF2
SCHEMBL8032174 0.76 F2 (0.58) ACSL1RORCBCHECNR2F2
SCHEMBL8015782 0.76 RORC (0.58) RORCHDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1060166-A1 FIVE-MEMBERED, BENZO-CONDENSED HETEROCYCLES USED AS ANTITHROMBOTIC AGENTS Boehringer Ingelheim Pharma KG (DE) 2000-12-20 EP disclosed
US-6114532-A ANTICOAGULANT BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-05 US disclosed
WO-1999040072-A1 FIVE-MEMBERED, BENZO-CONDENSED HETEROCYCLES USED AS ANTITHROMBOTIC AGENTS BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-08-12 WO disclosed