SCHEMBL8032987

SCHEMBL8032987

CNc1ccc(C2(C(=O)O)CC2)cc1N

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKCI P41743 1/20 0.53
AKR1C3 P42330 5/20 0.44
AKR1C2 P52895 5/20 0.44
AKR1C1 Q04828 4/20 0.44
AKR1B10 O60218 1/20 0.44
AKR1C4 P17516 1/20 0.44
APP P05067 6/20 0.43
CYP2C19 P33261 5/20 0.43
CYP3A4 P08684 5/20 0.43
CYP2C9 P11712 4/20 0.43
CYP2D6 P10635 2/20 0.43
PSEN1 P49768 1/20 0.41
PSEN2 P49810 1/20 0.41
APH1B Q8WW43 1/20 0.41
NCSTN Q92542 1/20 0.41
APH1A Q96BI3 1/20 0.41
PSENEN Q9NZ42 1/20 0.41
TLR7 Q9NYK1 1/20 0.37
HDAC3 O15379 1/20 0.37
NCOR2 Q9Y618 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12846569 0.83 AKR1C3 (0.43) PRKCIAKR1C3AKR1C2AKR1C1AKR1B10
SCHEMBL7412365 0.80 PRKCI (0.42) PRKCICYP3A4HDAC3
SCHEMBL7410812 0.80 HSD11B1 (0.52) PRKCICYP2C19CYP3A4CYP2C9HDAC3
SCHEMBL2450173 0.77 APP (0.47) AKR1C3AKR1C2AKR1C1AKR1B10AKR1C4
SCHEMBL12846323 0.77 AKR1C3 (0.40) AKR1C3AKR1C2AKR1C1AKR1B10AKR1C4
SCHEMBL7412565 0.77 HCAR3 (0.57) AKR1C3AKR1C2AKR1C1AKR1B10AKR1C4
SCHEMBL7415701 0.76 HDAC1 (0.41) PRKCIHDAC3
SCHEMBL7980982 0.74 OPRM1 (0.45)
SCHEMBL21968864 0.71 AKR1C1 (0.49) AKR1C3AKR1C2AKR1C1AKR1B10AKR1C4
SCHEMBL23250799 0.71 AKR1C1 (0.39) AKR1C3AKR1C2AKR1C1APPCYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114532-A ANTICOAGULANT BOEHRINGER INGELHEIM PHARMA KG (DE) 2000-09-05 US disclosed