SCHEMBL8033656

SCHEMBL8033656

CC(C)(C)c1ccc(-n2nnnc2Sc2ncc(C(=O)O)s2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.41
HTT P42858 5/20 0.41
KMT2A Q03164 5/20 0.41
MAPT P10636 5/20 0.41
LMNA P02545 3/20 0.41
TP53 P04637 2/20 0.41
MAPK1 P28482 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
HSD17B10 Q99714 2/20 0.41
HPGD P15428 4/20 0.40
RECQL P46063 1/20 0.39
EP300 Q09472 1/20 0.37
MEN1 O00255 3/20 0.37
POLB P06746 3/20 0.37
KDM4E B2RXH2 2/20 0.36
PKM P14618 2/20 0.36
TSHR P16473 2/20 0.36
HCAR2 Q8TDS4 1/20 0.36
RXRA P19793 1/20 0.36
RXRB P28702 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8045818 0.86 HPGD (0.51) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL8044465 0.86 ALDH1A1 (0.51) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL8046081 0.86 ALDH1A1 (0.46) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL8042658 0.85 KMT2A (0.42) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL8033822 0.85 KDM4E (0.54) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL8047631 0.85 MAPT (0.41) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL8044703 0.82 MAPT (0.44) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL8048031 0.82 PTGS2 (0.45) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL8042810 0.81 ALDH1A1 (0.43) ALDH1A1HTTKMT2AMAPTLMNA
SCHEMBL8042077 0.80 ALDH1A1 (0.39) ALDH1A1HTTKMT2AMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed