SCHEMBL8034221

SCHEMBL8034221

COC(=O)C(=Cc1ccc(Cl)c(C(F)(F)F)c1)C(C)=O

nearest known ligand 0.49

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NPFFR1 Q9GZQ6 2/20 0.45
NPFFR2 Q9Y5X5 2/20 0.45
GAA P10253 2/20 0.43
KDR P35968 2/20 0.43
TDP1 Q9NUW8 1/20 0.43
NOTUM Q6P988 2/20 0.42
MAPT P10636 2/20 0.42
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
LMNA P02545 1/20 0.41
KDM4E B2RXH2 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8120081 1.00 NPFFR1 (0.45) NPFFR1NPFFR2GAAKDRTDP1
SCHEMBL8879892 0.90 GAA (0.43) GAATDP1MAPTKDM4E
SCHEMBL8879894 0.90 GAA (0.43) GAATDP1MAPTKDM4E
SCHEMBL29079163 0.85 GAA (0.44) GAATDP1MAPT
SCHEMBL8997541 0.85 NPFFR2 (0.45) NPFFR1NPFFR2GAAKDRTDP1
SCHEMBL8997535 0.85 NPFFR2 (0.45) NPFFR1NPFFR2GAAKDRTDP1
SCHEMBL28449048 0.83 GAA (0.50) GAATDP1MAPTKDM4E
SCHEMBL3311082 0.80 NPFFR1 (0.43) NPFFR1NPFFR2GAAKDRNOTUM
SCHEMBL8880883 0.77 ALDH1A1 (0.46) GAATDP1HDAC1HDAC8HDAC6
SCHEMBL8880889 0.77 ALDH1A1 (0.46) GAATDP1HDAC1HDAC8HDAC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0891322-B1 DIMETHYL-SUBSTITUTED CYCLOHEXANE DIENE DERIVATIVES BAYER AG (DE) 2000-12-27 EP disclosed
US-6103925-A MUSCLE CONTRACTION INHIBITORS; MODULATOR WITH SELECTIVITY FOR CHARYBDOTOXIN-SENSITIVE, CALCIUM-DEPENDENT POTASSIUM CHANNELS BAYER AKTIENGESELLSCHAFT (DE) 2000-08-15 US disclosed
EP-0758648-B1 Substituted 4H-pyrans with a modulating effect on calcium channels BAYER AG (DE) 2000-03-15 EP disclosed
US-5760073-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS BAYER AKTIENGESELLSCHAFT (DE) 1998-06-02 US disclosed
EP-0758648-A1 Substituted 4H-pyrans with a modulating effect on calcium channels BAYER AG (DE) 1997-02-19 EP disclosed