SCHEMBL8035149

SCHEMBL8035149

CCCN(CCC)C(=O)NC(=O)c1c(C(F)(F)F)cc(OC)c(O)c1[N+](=O)[O-]

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.36
CYP3A4 P08684 2/20 0.34
TDP1 Q9NUW8 2/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP2C19 P33261 2/20 0.34
MAPT P10636 2/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
ALOX12 P18054 1/20 0.34
ALDH1A1 P00352 3/20 0.33
KMT2A Q03164 3/20 0.33
MEN1 O00255 2/20 0.33
CYP1A2 P05177 1/20 0.33
KDM4E B2RXH2 2/20 0.32
POLB P06746 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
CTDSP1 Q9GZU7 1/20 0.32
LRRK2 Q5S007 1/20 0.32
PRMT5 O14744 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8035726 0.94 CYP3A4 (0.35) NPSR1CYP3A4TDP1TSHRMAPK1
SCHEMBL8035145 0.92 LRRK2 (0.35) CYP3A4TDP1CYP2C19MAPTCYP2D6
SCHEMBL8025556 0.85 NPSR1 (0.42) NPSR1CYP3A4TDP1CYP2C19MAPT
SCHEMBL8037862 0.82 CYP3A4 (0.38) NPSR1CYP3A4TDP1TSHRMAPK1
SCHEMBL8034312 0.80 TBXA2R (0.38)
SCHEMBL8038463 0.80 EPHX2 (0.39)
SCHEMBL8036201 0.80 EPHX2 (0.39)
SCHEMBL8028327 0.80 POLB (0.37) NPSR1MAPK1CYP2C19MAPTCYP2D6
SCHEMBL8040235 0.78 CYP3A4 (0.30) CYP3A4TDP1TSHRMAPK1
SCHEMBL8023142 0.78 ALDH1A1 (0.39) CYP3A4CYP2C19MAPTALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed