SCHEMBL8023142

SCHEMBL8023142

CCOCCNC(=O)NC(=O)c1c(C(F)(F)F)cc(OC)c(O)c1[N+](=O)[O-]

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
KMT2A Q03164 5/20 0.39
MEN1 O00255 3/20 0.39
NPC1 O15118 2/20 0.39
MAPT P10636 2/20 0.39
KDM4E B2RXH2 1/20 0.39
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C19 P33261 1/20 0.35
POLB P06746 3/20 0.35
LMNA P02545 2/20 0.33
TP53 P04637 1/20 0.33
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LRRK2 Q5S007 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8037015 0.94 ALDH1A1 (0.45) ALDH1A1KMT2AMEN1NPC1MAPT
SCHEMBL8041408 0.89 SMN1; SMN2 (0.32) ALDH1A1KMT2AMEN1NPC1MAPT
SCHEMBL8034312 0.88 TBXA2R (0.38)
SCHEMBL8036201 0.87 EPHX2 (0.39)
SCHEMBL8038463 0.87 EPHX2 (0.39)
SCHEMBL8035145 0.79 LRRK2 (0.35) ALDH1A1KMT2AMEN1MAPTKDM4E
SCHEMBL8025559 0.79 MAPT (0.37) ALDH1A1KMT2AMAPTKDM4ECYP2C19
SCHEMBL8035149 0.78 NPSR1 (0.36) ALDH1A1KMT2AMEN1MAPTKDM4E
SCHEMBL8022533 0.77 G6PD (0.38) KMT2AMEN1NPC1MAPTCYP3A4
SCHEMBL8035132 0.77 S1PR1 (0.38) KMT2AMEN1KDM4ETP53LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed