SCHEMBL8037862

SCHEMBL8037862

CCCCN(CCCC)C(=O)NC(=O)c1c(C(F)(F)F)cc(O)c(O)c1[N+](=O)[O-]

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.38
MAPK1 P28482 2/20 0.38
MAPT P10636 2/20 0.38
COMT P21964 3/20 0.36
TSHR P16473 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
HTT P42858 2/20 0.32
LMNA P02545 1/20 0.31
VCAM1 P19320 1/20 0.31
UBE2M P61081 1/20 0.31
DCUN1D1 Q96GG9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8035726 0.88 CYP3A4 (0.35) CYP3A4MAPK1MAPTTSHRTDP1
SCHEMBL8040235 0.84 CYP3A4 (0.30) CYP3A4MAPK1TSHRTDP1
SCHEMBL8035149 0.82 NPSR1 (0.36) CYP3A4MAPK1MAPTTSHRTDP1
SCHEMBL8035781 0.80 EPHX2 (0.41)
SCHEMBL8041445 0.80 EPHX2 (0.41)
SCHEMBL8035145 0.77 LRRK2 (0.35) CYP3A4MAPTCOMTTDP1ALDH1A1
SCHEMBL8035603 0.76 RAB9A (0.40) MAPTALDH1A1SMN1; SMN2NPSR1
SCHEMBL8035695 0.74 COMT (0.32) COMT
SCHEMBL8035622 0.74 COMT (0.37) MAPK1MAPTCOMTALDH1A1SMN1; SMN2
SCHEMBL8041408 0.73 SMN1; SMN2 (0.32) MAPK1MAPTCOMTALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed