SCHEMBL8035623

SCHEMBL8035623

COc1cc(C(F)(F)F)c(C(=O)NC(=O)Nc2ccccc2C(C)(C)C)cc1OCc1ccccc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.47
LPAR1 Q92633 1/20 0.46
S1PR1 P21453 6/20 0.46
CTSV O60911 2/20 0.44
CTSL P07711 2/20 0.44
SMPD1 P17405 1/20 0.42
HDAC1 Q13547 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
BRD4 O60885 1/20 0.41
LMNA P02545 2/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ADRB2 P07550 1/20 0.41
GPR183 P32249 1/20 0.41
APLNR P35414 1/20 0.41
S1PR5 Q9H228 1/20 0.41
POLB P06746 2/20 0.41
PKM P14618 1/20 0.41
KDM4E B2RXH2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8035613 0.88 S1PR1 (0.54) S1PR1CTSVCTSLSMPD1HDAC1
SCHEMBL8025544 0.85 ALDH1A1 (0.49) S1PR1CTSVCTSLSMPD1HDAC1
SCHEMBL8035621 0.84 ATM (0.48) S1PR1CTSVCTSLSMPD1HDAC1
SCHEMBL8025540 0.84 SMN1; SMN2 (0.48) S1PR1CTSVCTSLSMPD1HDAC1
SCHEMBL8040248 0.83 MTNR1A (0.52) S1PR1CTSVCTSLSMPD1HDAC1
SCHEMBL8037334 0.83 S1PR1 (0.43) S1PR1CTSVCTSLSMPD1HDAC1
SCHEMBL8039098 0.83 HPGD (0.48) S1PR1CTSVCTSLSMPD1HDAC1
SCHEMBL8039086 0.82 MTNR1A (0.47) S1PR1CTSVCTSLSMPD1HDAC1
SCHEMBL8037331 0.81 MTNR1A (0.46) S1PR1SMPD1HDAC1HDAC8HDAC6
SCHEMBL8025483 0.81 MEN1 (0.46) S1PR1CTSVCTSLSMPD1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed