SCHEMBL8025544

SCHEMBL8025544

COc1cc(C(F)(F)F)c(C(=O)NC(=O)NC(C)(C)C)cc1OCc1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
HPGD P15428 3/20 0.49
KDM4E B2RXH2 2/20 0.49
SMPD1 P17405 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
S1PR1 P21453 3/20 0.45
CTSV O60911 2/20 0.44
CTSL P07711 2/20 0.44
LMNA P02545 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.42
MAPK1 P28482 1/20 0.42
HTT P42858 1/20 0.42
NPC1 O15118 2/20 0.42
RAB9A P51151 1/20 0.42
MRGPRX4 Q96LA9 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SRD5A1 P18405 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8035613 0.88 S1PR1 (0.54) ALDH1A1HPGDKDM4ESMPD1HDAC1
SCHEMBL8039098 0.87 HPGD (0.48) ALDH1A1HPGDKDM4ESMPD1HDAC1
SCHEMBL8025540 0.86 SMN1; SMN2 (0.48) ALDH1A1HPGDKDM4ESMPD1HDAC1
SCHEMBL8035623 0.85 IDO1 (0.47) KDM4ESMPD1HDAC1HDAC8HDAC6
SCHEMBL8041285 0.85 ALDH1A1 (0.51) ALDH1A1HPGDKDM4ESMPD1HDAC1
SCHEMBL8025483 0.85 MEN1 (0.46) ALDH1A1SMPD1HDAC1HDAC8HDAC6
SCHEMBL8040248 0.85 MTNR1A (0.52) ALDH1A1HPGDKDM4ESMPD1HDAC1
SCHEMBL8037334 0.85 S1PR1 (0.43) ALDH1A1HPGDKDM4ESMPD1HDAC1
SCHEMBL8037062 0.85 SMPD1 (0.51) ALDH1A1HPGDKDM4ESMPD1HDAC1
SCHEMBL8025476 0.84 SMPD1 (0.47) HPGDKDM4ESMPD1HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed