SCHEMBL8035910

SCHEMBL8035910

C=CCCNCc1ccc(-c2ccc(C(=O)c3ccc(C#N)cc3)cc2)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 6/20 0.46
PPARA Q07869 2/20 0.42
KDM1A O60341 1/20 0.42
HDAC1 Q13547 1/20 0.42
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA4 P22748 1/20 0.41
CA9 Q16790 1/20 0.41
EPHX2 P34913 1/20 0.41
SAE1 Q9UBE0 1/20 0.39
UBA2 Q9UBT2 1/20 0.39
LOXL2 Q9Y4K0 1/20 0.39
AKR1C3 P42330 1/20 0.39
LSS P48449 1/20 0.38
SCN8A Q9UQD0 1/20 0.38
CD274 Q9NZQ7 1/20 0.37
NAMPT P43490 1/20 0.37
HDAC2 Q92769 1/20 0.37
CNR1 P21554 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9442705 0.99 VNN1 (0.45) VNN1PPARAKDM1AHDAC1CA12
SCHEMBL9150945 0.83 LSS (0.40) VNN1HDAC1LSS
SCHEMBL9149679 0.83 LSS (0.54) HDAC1CA12CA1CA2CA4
Hydrochloric Acid SCHEMBL9442716 0.82 S1PR1 (0.45) VNN1PPARAHDAC1LSSHDAC2
SCHEMBL3675152 0.79 SRD5A2 (0.44) HDAC1EPHX2LSS
Hydrochloric Acid SCHEMBL9442719 0.77 ACHE (0.45) HDAC1HDAC2
SCHEMBL8904444 0.76 PLK1 (0.47) HDAC1EPHX2HDAC2
SCHEMBL9442728 0.76 CHRNA7 (0.42) PPARAHDAC1HDAC2
SCHEMBL8046483 0.76 LSS (0.44) VNN1LSS
Hydrochloric Acid SCHEMBL8902724 0.75 CHRNA7 (0.41) PPARAHDAC1HDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636367-B1 Use of phenylalkylamines for producing cholesterol lowering agents HOFFMANN LA ROCHE (CH) 2000-03-29 EP claimed
US-5574071-A ADMINISTERING PHENYLALKYLAMINO KETONES HOFFMANN-LA ROCHE INC. (US) 1996-11-12 US claimed
EP-0636367-A1 Use of phenylalkylamines for producing cholesterol lowering agents F. HOFFMANN-LA ROCHE AG (CH) 1995-02-01 EP claimed
EP-0636367-B1 Use of phenylalkylamines for producing cholesterol lowering agents HOFFMANN LA ROCHE (CH) 2000-03-29 EP disclosed
US-5637771-A Compound useful for lowering cholesterol HOFFMANN-LA ROCHE INC. (US) 1997-06-10 US disclosed
US-5574071-A ADMINISTERING PHENYLALKYLAMINO KETONES HOFFMANN-LA ROCHE INC. (US) 1996-11-12 US disclosed
US-5495048-A ANTICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
EP-0636367-A1 Use of phenylalkylamines for producing cholesterol lowering agents F. HOFFMANN-LA ROCHE AG (CH) 1995-02-01 EP disclosed