SCHEMBL8035926

SCHEMBL8035926

CC(C)(C)OC(=O)N[C@H](N)Cc1ccc(-c2ccc(C#N)c(F)c2)cc1

nearest known ligand 0.53

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.53
CTSK P43235 8/20 0.49
CTSS P25774 8/20 0.49
CTSC P53634 8/20 0.46
EGLN2 Q96KS0 1/20 0.46
PTPN1 P18031 1/20 0.45
CTSB P07858 2/20 0.45
GPR119 Q8TDV5 1/20 0.44
CTSL P07711 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22046325 0.88 CTSC (0.58) TRPA1CTSKCTSSCTSCEGLN2
SCHEMBL12383142 0.88 CTSC (0.58) TRPA1CTSKCTSSCTSCEGLN2
SCHEMBL8036118 0.82 CTSS (0.55) CTSKCTSSCTSCPTPN1CTSB
SCHEMBL21266172 0.81 TRPA1 (0.50) TRPA1CTSKCTSSCTSCEGLN2
SCHEMBL30751838 0.81 TRPA1 (0.50) TRPA1CTSKCTSSCTSCEGLN2
SCHEMBL8031921 0.79 GPR119 (0.47) CTSKCTSCGPR119
SCHEMBL536951 0.78 CTSC (0.50) CTSKCTSC
SCHEMBL27669003 0.78 EGLN2 (0.62) TRPA1EGLN2GPR119
SCHEMBL25152842 0.78 TRPA1 (0.56) TRPA1CTSKCTSSEGLN2PTPN1
SCHEMBL21639072 0.78 CTSS (0.57) TRPA1CTSKCTSSPTPN1CTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009074829-A1 PEPTIDYL NITRILES AND USE THEREOF AS DIPEPTIDYL PEPTIDASE I INHIBITORS ASTRAZENECA AB (SE) 2009-06-18 WO disclosed