SCHEMBL8035971

SCHEMBL8035971

O=c1oc2cc3oc(=O)sc3cc2s1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOA P21397 6/20 0.57
MAOB P27338 6/20 0.57
MAPT P10636 4/20 0.57
ALPI P09923 2/20 0.57
ALPG P10696 2/20 0.57
HPGD P15428 2/20 0.57
HTT P42858 2/20 0.57
CA2 P00918 1/20 0.57
CUL4A Q13619 4/20 0.45
GAA P10253 4/20 0.41
PKM P14618 3/20 0.41
KMT2A Q03164 4/20 0.39
ALDH1A1 P00352 3/20 0.39
POLB P06746 3/20 0.39
KDM4E B2RXH2 4/20 0.37
HSD17B10 Q99714 4/20 0.37
TDP1 Q9NUW8 4/20 0.37
ALOX15 P16050 3/20 0.37
ALOX12 P18054 3/20 0.37
ALPL P05186 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11637378 0.78 MAOA (0.52) MAOAMAOBMAPTALPIALPG
SCHEMBL6002101 0.75 CUL4A (0.54) MAOAMAOBMAPTALPIALPG
SCHEMBL6001543 0.75 CUL4A (0.54) MAOAMAOBMAPTALPIALPG
SCHEMBL5541064 0.75 MAOA (0.63) MAOAMAOBMAPTALPIALPG
SCHEMBL995285 0.73 MAPT (0.47) MAOAMAOBMAPTALPIALPG
Tioxolone SCHEMBL36433 0.73 MAOA (1.00) MAOAMAOBMAPTALPIALPG
SCHEMBL2056163 0.73 MAOA (0.61) MAOAMAOBMAPTALPIALPG
SCHEMBL995283 0.73 MAPT (0.47) MAOAMAOBMAPTALPIALPG
SCHEMBL10397843 0.71 MAPT (0.49) MAOAMAOBMAPTALPIALPG
SCHEMBL3802319 0.69 MAOA (0.58) MAOAMAOBMAPTALPIALPG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0832054-B1 HETEROCYCLIC METHYL FREE RADICALS AS IMAGE ENHANCING AGENTS NYCOMED IMAGING AS (NO) 2000-12-27 EP disclosed
US-6063360-A USEFUL AS CONTRAST AGENT FOR OVERHAUSER MAGNETIC RESONACE IMAGING NYCOMED IMAGING A/S (NO) 2000-05-16 US disclosed
EP-0662004-B1 USE OF PERSISTENT FREE-RADICALS IN MAGNETIC RESONANCE IMAGING NYCOMED INNOVATION AB (SE) 1998-03-18 EP disclosed
WO-1996039367-A1 HETEROCYCLIC METHYL FREE RADICALS AS IMAGE ENHANCING AGENTS NYCOMED IMAGING A/S (NO) 1996-12-12 WO disclosed
US-5530140-A Free radicals NYCOMED IMAGING AS (NO) 1996-06-25 US disclosed
US-5435991-A Use of persistent heterocyclic free-radicals in magnetic resonance imaging NYCOMED INNOVATION AB (SE) 1995-07-25 US disclosed
EP-0662004-A1 USE OF PERSISTENT FREE-RADICALS IN MAGNETIC RESONANCE IMAGING Nycomed Innovation AB (SE) 1995-07-12 EP disclosed
WO-1993002711-A1 USE OF PERSISTENT FREE-RADICALS IN MAGNETIC RESONANCE IMAGING NYCOMED INNOVATION AB (SE) 1993-02-18 WO disclosed