SCHEMBL8038722

SCHEMBL8038722

O=S(=O)(c1ccccc1)N(SCl)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
APOBEC3G Q9HC16 1/20 0.47
ALDH1A1 P00352 2/20 0.46
PKM P14618 1/20 0.46
ESR1 P03372 3/20 0.43
KMT2A Q03164 2/20 0.42
CA12 O43570 1/20 0.42
CA9 Q16790 1/20 0.42
TDP1 Q9NUW8 2/20 0.41
HSD17B10 Q99714 2/20 0.41
LMNA P02545 1/20 0.40
HTR6 P50406 1/20 0.39
HSD11B1 P28845 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8038717 0.88 CA12 (0.60) ALDH1A1PKMKMT2ACA12CA9
SCHEMBL8028854 0.80 APOBEC3G (0.47) APOBEC3GALDH1A1PKMESR1KMT2A
SCHEMBL4828287 0.79 CDK1 (0.43) APOBEC3GALDH1A1PKMESR1KMT2A
SCHEMBL18421807 0.79 ALDH1A1 (0.46) APOBEC3GALDH1A1PKMESR1KMT2A
SCHEMBL27951833 0.79 CDK1 (0.43) APOBEC3GALDH1A1PKMESR1KMT2A
SCHEMBL25238002 0.79 APOBEC3G (0.42) APOBEC3GALDH1A1PKMESR1KMT2A
SCHEMBL8039423 0.78 MEN1 (0.40) ALDH1A1PKMKMT2ACA12CA9
SCHEMBL18421903 0.77 ALDH1A1 (0.40) APOBEC3GALDH1A1PKMESR1KMT2A
SCHEMBL18421901 0.75 ALDH1A1 (0.39) APOBEC3GALDH1A1PKMESR1KMT2A
SCHEMBL18421900 0.74 ALDH1A1 (0.38) APOBEC3GALDH1A1PKMESR1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 47 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5756590-A MIXING TERPOLYMER WITH HALOTHIOSULFONAMIDE AND INCLUDING A HYDROHALIC ACID ACCEPTOR; OZONE RESISTANT TIRE SIDEWALLS THE GOODYEAR TIRE & RUBBER COMPANY (US) 1998-05-26 US claimed
EP-0312484-B1 Modification process GOODYEAR TIRE & RUBBER (US) 1993-11-24 EP claimed
EP-0377552-B1 PROCESS FOR SYNTHESIZING N-CHLOROTHIO-SULFONAMIDES THE GOODYEAR TIRE & RUBBER COMPANY (US) 1993-07-28 EP claimed
US-5187240-A Treatment of polyolefin polymer with N-halothiosulfonamide EXXON CHEMICAL PATENTS INC. (US) 1993-02-16 US claimed
US-5037896-A Selective catalytic process for preparing N-halothiosulfonamide modified polyolefins EXXON CHEMICAL PATENTS INC. (US) 1991-08-06 US claimed
US-5034467-A For polymers of high tensile strength EXXON CHEMICAL PATENTS, INC. (US) 1991-07-23 US claimed
US-5034468-A For polymers of high tensile strength EXXON CHEMICAL PATENTS INC. (US) 1991-07-23 US claimed
US-4992583-A Reacting n,n'-dithiobis (sulfonamide) with chlorine gas or sulfuryl chloride THE GOODYEAR TIRE & RUBBER COMPANY (US) 1991-02-12 US claimed
US-4956420-A USING A COPPER, ANTIMONY, BISMITH OR TIN SALT OF AN ORGANIC MONO-OR POLYCARBOXYLIC ACID EXXON CHEMICAL PATENTS INC. (US) 1990-09-11 US claimed
EP-0377552-A1 Process for synthesizing N-chlorothio-sulfonamides THE GOODYEAR TIRE & RUBBER COMPANY (US) 1990-07-11 EP claimed
US-4910266-A Modification process using N-chloro-thiosulfonamide and rubber THE GOODYEAR TIRE & RUBBER COMPANY (US) 1990-03-20 US claimed
US-4820780-A Modification of rubber with N-chlorothio-sulfonamide THE GOODYEAR TIRE & RUBBER COMPANY (US) 1989-04-11 US claimed
US-4617347-A CONVEYOR BELTS THE GOODYEAR TIRE & RUBBER COMPANY (US) 1986-10-14 US claimed
EP-0989171-A1 N-halothio-amide-modified elastomers and their application as adhesives for precured elastomeric substrates THE GOODYEAR TIRE & RUBBER COMPANY (US) 2000-03-29 EP disclosed
EP-0733651-B1 Process for preparation of N-halothiosulfonamide modified terpolymers GOODYEAR TIRE & RUBBER (US) 1999-09-01 EP disclosed
US-5756590-A MIXING TERPOLYMER WITH HALOTHIOSULFONAMIDE AND INCLUDING A HYDROHALIC ACID ACCEPTOR; OZONE RESISTANT TIRE SIDEWALLS THE GOODYEAR TIRE & RUBBER COMPANY (US) 1998-05-26 US disclosed
US-4804028-A Non-staining vulcanized elastomeric composition and tires having sidewalls comprising said composition THE GOODYEAR TIRE & RUBBER COMPANY (US) 1989-02-14 US disclosed
EP-0240448-A2 Non-staining vulcanized elastomeric composition and tires having sidewalls comprising said composition THE GOODYEAR TIRE & RUBBER COMPANY (US) 1987-10-07 EP disclosed
US-4617347-A CONVEYOR BELTS THE GOODYEAR TIRE & RUBBER COMPANY (US) 1986-10-14 US disclosed
US-3970133-A Chlorothio-sulfonamide-modified rubbery terpolymers and their blends THE GOODYEAR TIRE & RUBBER COMPANY (US) 1976-07-20 US disclosed