SCHEMBL8039587

SCHEMBL8039587

NC(=O)CCCCCCN(C(=O)OCc1ccccc1)C(N)=NC(=O)OCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR6 P51684 1/20 0.42
PAX8 Q06710 1/20 0.42
ALDH1A1 P00352 3/20 0.36
HDAC3 O15379 2/20 0.36
NCOR2 Q9Y618 2/20 0.36
MAPK1 P28482 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35
KMT2A Q03164 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
HTT P42858 1/20 0.35
LTA4H P09960 1/20 0.35
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
ALOX5 P09917 1/20 0.34
SIRT2 Q8IXJ6 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL989683 0.95 CCR6 (0.45) CCR6PAX8ALDH1A1MAPK1L3MBTL1
SCHEMBL8029844 0.94 HTT (0.42) CCR6PAX8ALDH1A1HDAC3NCOR2
SCHEMBL7242187 0.94 HTT (0.42) CCR6PAX8ALDH1A1HDAC3NCOR2
SCHEMBL7352897 0.93 HTT (0.43) CCR6PAX8ALDH1A1HDAC3MAPK1
SCHEMBL6661417 0.89 CCR6 (0.41) CCR6PAX8ALDH1A1MAPK1L3MBTL1
SCHEMBL7359299 0.89 HTT (0.44) CCR6PAX8ALDH1A1HDAC3MAPK1
SCHEMBL7355382 0.86 HTT (0.43) CCR6PAX8ALDH1A1MAPK1L3MBTL1
SCHEMBL7358565 0.84 CCR6 (0.39) CCR6PAX8ALDH1A1MAPK1L3MBTL1
SCHEMBL6827318 0.84 CTSL (0.39) CCR6PAX8ALDH1A1MAPK1L3MBTL1
SCHEMBL9228435 0.81 ALDH1A1 (0.41) CCR6PAX8ALDH1A1MAPK1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0765866-B1 Preparation of optically active (S)-(-) and (R)-(+)- deoxyspergualin and novel intermediates thereof BRISTOL MYERS SQUIBB CO (US) 2000-12-06 EP disclosed
US-5869734-A Preparation of optically active (S)-(-) and (R)-(+)-deoxyspergualin and novel intermediates thereof BRISTOL-MYERS SQUIBB CO. (US) 1999-02-09 US disclosed
EP-0765866-A2 Preparation of optically active (S)-(-) and (R)-(+)- deoxyspergualin and novel intermediates thereof BRISTOL-MYERS SQUIBB COMPANY (US) 1997-04-02 EP disclosed