SCHEMBL8040147

SCHEMBL8040147

N#Cc1nc2cccc(O)c2s1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PSMB8 P28062 2/20 0.67
APP P05067 1/20 0.46
ACHE P22303 1/20 0.41
SOS2 Q07890 1/20 0.40
GSK3A P49840 4/20 0.39
GSK3B P49841 4/20 0.39
CCNB2 O95067 1/20 0.39
CDK1 P06493 1/20 0.39
CCNB1 P14635 1/20 0.39
CDK5 Q00535 1/20 0.39
CDK5R1 Q15078 1/20 0.39
CCNB3 Q8WWL7 1/20 0.39
ALDH1A1 P00352 3/20 0.37
KMT2A Q03164 3/20 0.37
MAPT P10636 2/20 0.37
NPSR1 Q6W5P4 2/20 0.37
GAA P10253 1/20 0.37
RAB9A P51151 1/20 0.37
CA2 P00918 1/20 0.34
PDPK1 O15530 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21063750 0.80 PSMB8 (0.65) PSMB8GSK3AGSK3BCCNB2CDK1
SCHEMBL8034068 0.77 PSMB8 (0.49) PSMB8GSK3AGSK3BCCNB2CDK1
SCHEMBL8022630 0.77 PSMB8 (0.57) PSMB8GSK3AGSK3BCCNB2CDK1
SCHEMBL24256511 0.76 PSMB8 (0.59) PSMB8GSK3AGSK3BCCNB2CDK1
SCHEMBL10574548 0.73 PSMB8 (0.65) PSMB8APPACHESOS2ALDH1A1
SCHEMBL1046142 0.72 PSMB8 (0.43) PSMB8GSK3AGSK3BCCNB2CDK1
SCHEMBL30938811 0.71 PSMB8 (0.53) PSMB8ALDH1A1KMT2AMAPTGAA
SCHEMBL492446 0.71 PSMB8 (0.53) PSMB8ALDH1A1KMT2AMAPTGAA
SCHEMBL9305472 0.71 APP (0.46) PSMB8APPACHEALDH1A1KMT2A
SCHEMBL9305900 0.71 APP (0.46) PSMB8APPACHEALDH1A1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6130217-A ANTITUMOR PFIZER INC (US) 2000-10-10 US disclosed
WO-1994022846-A1 COMPOUNDS ENHANCING ANTITUMOR ACTIVITY OF OTHER CYTOTOXIC AGENTS PFIZER INC. (US) 1994-10-13 WO disclosed