SCHEMBL8040804

SCHEMBL8040804

Cc1cc(C(O)=CC(=O)C(=O)O)ccc1Cl

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.50
CA12 O43570 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
CA9 Q16790 1/20 0.50
TAS1R3 Q7RTX0 1/20 0.43
TAS1R1 Q7RTX1 1/20 0.43
TAS1R2 Q8TE23 1/20 0.43
PTPN1 P18031 1/20 0.42
MAOA P21397 1/20 0.42
MAOB P27338 1/20 0.42
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
MCL1 Q07820 1/20 0.41
TSHR P16473 2/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
S1PR3 Q99500 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8040803 1.00 CYP1A2 (0.50) CYP1A2CA12CA1CA2CA9
SCHEMBL8369833 0.84 ALDH1A1 (0.63) CA12CA1CA2CA9TAS1R3
SCHEMBL8369834 0.84 ALDH1A1 (0.63) CA12CA1CA2CA9TAS1R3
SCHEMBL8040827 0.84 CA12 (0.55) CYP1A2CA12CA1CA2CA9
SCHEMBL8046164 0.84 TSHR (0.57) CYP1A2CA12CA1CA2CA9
SCHEMBL8046161 0.84 TSHR (0.57) CYP1A2CA12CA1CA2CA9
SCHEMBL8040833 0.84 CA12 (0.55) CYP1A2CA12CA1CA2CA9
SCHEMBL5902813 0.82 ALDH1A1 (0.46) CYP1A2TAS1R3TAS1R1TAS1R2PTPN1
SCHEMBL5902812 0.82 ALDH1A1 (0.46) CYP1A2TAS1R3TAS1R1TAS1R2PTPN1
SCHEMBL7845572 0.77 TAS1R3 (0.49) CYP1A2TAS1R3TAS1R1TAS1R2MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0868420-B1 3-PYRAZOLECARBOXAMIDE DERIVATIVES HAVING CANNABINOID RECEPTOR AFFINITY SANOFI SYNTHELABO (FR) 2000-03-29 EP disclosed
EP-0885889-A2 Process for the preparation of pyrazole-3-carboxylic acids SANOFI (FR) 1998-12-23 EP disclosed