SCHEMBL8041268

SCHEMBL8041268

CCCN(C)C(=O)N(C)C(=O)c1c(Cl)cc(O)c(O)c1[N+](=O)[O-]

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
COMT P21964 9/20 0.40
VCAM1 P19320 3/20 0.33
ALDH1A1 P00352 2/20 0.33
HCAR3 P49019 1/20 0.32
MAPT P10636 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.31
CDK2 P24941 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8028100 0.86 L3MBTL1 (0.35) COMTALDH1A1MAPTL3MBTL1CDK2
SCHEMBL8037291 0.86 COMT (0.37) COMTALDH1A1MAPT
SCHEMBL8035686 0.82 COMT (0.38) COMTALDH1A1MAPTL3MBTL1CDK2
SCHEMBL8039069 0.81 COMT (0.40) COMTALDH1A1MAPT
SCHEMBL8041271 0.80 COMT (0.35) COMTALDH1A1MAPTL3MBTL1CDK2
SCHEMBL8037287 0.79 COMT (0.39) COMTALDH1A1MAPTL3MBTL1CDK2
SCHEMBL8044817 0.75 ALDH1A1 (0.35) VCAM1ALDH1A1MAPTL3MBTL1CDK2
SCHEMBL8035095 0.74 SPR (0.38) COMTALDH1A1MAPT
SCHEMBL7614112 0.73 COMT (0.43) COMTALDH1A1CDK2
SCHEMBL8039065 0.73 HSP90AA1 (0.47) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed