SCHEMBL8041763

SCHEMBL8041763

COc1cc(C(F)(F)F)c(C(=O)N(C)C(=O)N(C)C2CCCCC2)c([N+](=O)[O-])c1O

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
MAPT P10636 3/20 0.36
ALDH1A1 P00352 2/20 0.34
SMN1; SMN2 Q16637 2/20 0.34
MAPK1 P28482 1/20 0.34
NPSR1 Q6W5P4 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
POLB P06746 2/20 0.32
GAA P10253 1/20 0.32
CYP2D6 P10635 1/20 0.32
KDM4E B2RXH2 1/20 0.32
RAB9A P51151 1/20 0.32
AKR1C3 P42330 1/20 0.32
AKR1C1 Q04828 1/20 0.32
ERN1 O75460 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8041245 0.88 MAPT (0.39) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL8028327 0.84 POLB (0.37) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL8028359 0.82 SMN1; SMN2 (0.35) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL8041629 0.81 TDP1 (0.34) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL8038341 0.77 SMO (0.38) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL8040282 0.76 LRRK2 (0.33) ERN1
SCHEMBL8038220 0.75 PPIA (0.42) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL8028357 0.75 ALDH1A1 (0.41) MEN1KMT2AMAPTALDH1A1SMN1; SMN2
SCHEMBL8040084 0.74 ALDH1A1 (0.33) MAPTALDH1A1SMN1; SMN2NPSR1GAA
SCHEMBL8025559 0.71 MAPT (0.37) KMT2AMAPTALDH1A1SMN1; SMN2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed