SCHEMBL8041245

SCHEMBL8041245

CN(C(=O)c1c(C(F)(F)F)cc(O)c(O)c1[N+](=O)[O-])C(=O)N(C)C1CCCCC1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
MAPT P10636 2/20 0.39
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
POLB P06746 2/20 0.34
RAB9A P51151 2/20 0.34
ALDH1A1 P00352 2/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
HTT P42858 1/20 0.33
COMT P21964 1/20 0.32
KDM4E B2RXH2 1/20 0.32
NPC1 O15118 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8041763 0.88 MEN1 (0.37) MAPTMEN1KMT2APOLBRAB9A
SCHEMBL8035603 0.82 RAB9A (0.40) MAPTMEN1KMT2APOLBRAB9A
SCHEMBL8041249 0.80 TAS1R3 (0.35) ALDH1A1COMT
SCHEMBL8041271 0.79 COMT (0.35) MAPTMEN1KMT2APOLBRAB9A
SCHEMBL8035622 0.74 COMT (0.37) MAPTMEN1KMT2APOLBALDH1A1
SCHEMBL8025492 0.72 PPIA (0.49) MAPTMEN1KMT2ARAB9AALDH1A1
SCHEMBL8028327 0.71 POLB (0.37) MAPTMEN1KMT2APOLBRAB9A
SCHEMBL8035683 0.71 SMYD3 (0.32) COMT
SCHEMBL8040243 0.70 PPIA (0.47) MAPTMEN1KMT2ARAB9AALDH1A1
SCHEMBL8025508 0.70 ALDH1A1 (0.37) MAPTKMT2APOLBALDH1A1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009081892-A1 NOVEL CATECHOL DERIVATIVE, PHARMACEUTICAL COMPOSITION CONTAINING THE SAME, AND USE OF THOSE KISSEI PHARMACEUTICAL CO., LTD. (JP) 2009-07-02 WO disclosed