SCHEMBL8041784

SCHEMBL8041784

Cc1c(Cl)c(O)c(N)c(C(=O)O)c1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DPP4 P27487 1/20 0.36
LDHA P00338 2/20 0.35
LDHB P07195 2/20 0.35
KMT2A Q03164 2/20 0.34
KDM4E B2RXH2 1/20 0.34
ALDH1A1 P00352 2/20 0.33
MAPT P10636 2/20 0.33
TDP1 Q9NUW8 1/20 0.33
GAA P10253 1/20 0.33
MAPK1 P28482 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
DHODH Q02127 4/20 0.31
IMPDH2 P12268 1/20 0.31
CYP3A4 P08684 3/20 0.31
CYP1A2 P05177 1/20 0.31
CYP2C8 P10632 1/20 0.31
CYP2D6 P10635 1/20 0.31
CYP2A6 P11509 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8031083 0.88 DPP4 (0.36) DPP4LDHALDHBKMT2AKDM4E
SCHEMBL28840200 0.75 ALDH1A1 (0.40) DPP4LDHALDHBKMT2AKDM4E
SCHEMBL10618701 0.73 ALDH1A1 (0.39) DPP4LDHALDHBKMT2AKDM4E
SCHEMBL11654790 0.73 ALDH1A1 (0.41) DPP4LDHALDHBKMT2AKDM4E
SCHEMBL5589377 0.72 DPP4 (0.45) DPP4LDHALDHBKDM4EALDH1A1
SCHEMBL31643709 0.72 DPP4 (0.40) DPP4LDHALDHBKMT2AKDM4E
SCHEMBL14718570 0.72 DPP4 (0.45) DPP4LDHALDHBKMT2AKDM4E
SCHEMBL28055293 0.71 ALDH1A1 (0.40) DPP4LDHALDHBKMT2AKDM4E
SCHEMBL8041148 0.71 ALDH1A1 (0.38) DPP4ALDH1A1MAPTTDP1IMPDH2
SCHEMBL7577377 0.69 CES2 (0.41) DPP4KMT2AKDM4EALDH1A1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686144-B1 NEW COMPOUNDS UNIV MARYLAND (US) 2000-04-19 EP claimed
EP-0686144-B1 NEW COMPOUNDS UNIV MARYLAND (US) 2000-04-19 EP disclosed
US-5688945-A Compounds ASTRA AKTIEBOLAG (SE) 1997-11-18 US disclosed
US-5661183-A 3-hydroxy anthanilic acid derivatives THE UNIVERSITY OF MARYLAND (US) 1997-08-26 US disclosed
EP-0686144-A1 NEW COMPOUNDS Astra Aktiebolag (SE) 1995-12-13 EP disclosed
WO-1994019315-A1 NEW COMPOUNDS ASTRA AKTIEBOLAG (SE) 1994-09-01 WO disclosed