SCHEMBL8041854

SCHEMBL8041854

CC(C)(C)OC(=O)NN(C=O)CCCCCCCOc1ccc2c(c1)C(=N)c1ccccc1-2

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 5/20 0.42
CA12 O43570 5/20 0.38
CA1 P00915 5/20 0.38
CA2 P00918 5/20 0.38
CA9 Q16790 5/20 0.38
PTPN11 Q06124 1/20 0.36
MAOB P27338 5/20 0.36
MCHR1 Q99705 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8040104 0.87 KMT2A (0.43) PDK2CA12CA1CA2CA9
SCHEMBL8049234 0.76 MAPT (0.39) PDK2
SCHEMBL8046733 0.76 MAPT (0.39) PDK2
SCHEMBL8053515 0.76 MAPT (0.39) PDK2
SCHEMBL8052585 0.76 MAPT (0.39) PDK2
SCHEMBL8043998 0.75 MAPT (0.39) PDK2
SCHEMBL8052590 0.75 MAPT (0.39) PDK2
SCHEMBL8040111 0.71 PTPN11 (0.38) PDK2PTPN11
SCHEMBL8046738 0.70 HDAC1 (0.33)
SCHEMBL8052434 0.70 HDAC1 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009085978-A1 BRIDGED CARBOCYCLIC OXIME HEPATITIS C VIRUS SERINE PROTEASE INHIBITORS ENANTA PHARCEUTICALS, INC. (US) 2009-07-09 WO disclosed