SCHEMBL8042292

SCHEMBL8042292

C=CC(=O)C(C(C)=O)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TGM2 P21980 1/20 0.45
TEAD1 P28347 3/20 0.43
CES2 O00748 2/20 0.42
CES1 P23141 2/20 0.42
NR4A1 P22736 1/20 0.41
NR4A2 P43354 1/20 0.41
NR4A3 Q92570 1/20 0.41
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
GSK3B P49841 1/20 0.38
ACP3 P15309 1/20 0.37
FFAR1 O14842 3/20 0.37
AKR1C3 P42330 1/20 0.37
AKR1C2 P52895 1/20 0.37
EPHX2 P34913 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28470051 0.85 CYP1A2 (0.39) ALDH1A1CYP1A2FFAR1AKR1C3AKR1C2
SCHEMBL28224167 0.84 CES2 (0.39) TGM2TEAD1CES2ALDH1A1AKR1C3
SCHEMBL7252884 0.81 HDAC3 (0.42) TGM2CES2CES1ALDH1A1
SCHEMBL29090926 0.80 TEAD1 (0.48) TGM2TEAD1CES2CES1NR4A1
SCHEMBL4749899 0.80 CES2 (0.47) CES2CES1NR4A1NR4A2NR4A3
SCHEMBL7472615 0.80 CES2 (0.47) CES2CES1NR4A1NR4A2NR4A3
SCHEMBL8028836 0.80 ESR1 (0.43) ALDH1A1CYP1A2
SCHEMBL28468309 0.80 TGM2 (0.42) TGM2CES2CES1ALDH1A1
SCHEMBL28469749 0.78 BRD4 (0.50) CYP1A2
SCHEMBL8040582 0.75 MAPT (0.48) TGM2CES2CES1ALDH1A1ACP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0440324-B1 Substituted beta-diketones and their use in the treatment of inflammatory bowel disease ORION YHTYMAE OY (FI) 2000-04-12 EP claimed