SCHEMBL8042469

SCHEMBL8042469

COc1ccccc1C1CCN(CCCCN2C(=O)COc3ccccc32)C1

nearest known ligand 0.64

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 8/20 0.64
HTR2A P28223 3/20 0.64
MCHR1 Q99705 3/20 0.64
CHRM1 P11229 14/20 0.55
KCNH2 Q12809 5/20 0.50
CHRM2 P08172 1/20 0.50
CHRM4 P08173 1/20 0.50
CHRM5 P08912 1/20 0.50
CHRM3 P20309 1/20 0.50
ADRA1A P35348 1/20 0.50
HRH1 P35367 1/20 0.50
ADRA1B P35368 1/20 0.50
SMPD1 P17405 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8042466 1.00 DRD2 (0.64) DRD2HTR2AMCHR1CHRM1KCNH2
SCHEMBL8042446 0.84 GRIN1 (0.61) DRD2CHRM1CHRM2CHRM4CHRM5
SCHEMBL8042443 0.84 GRIN1 (0.61) DRD2CHRM1CHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL8045702 0.83 GRIN1 (0.60) DRD2CHRM1CHRM2CHRM4CHRM5
Hydrochloric Acid SCHEMBL8045698 0.83 GRIN1 (0.60) DRD2CHRM1CHRM2CHRM4CHRM5
SCHEMBL8042421 0.79 DRD2 (0.63) DRD2ADRA1AHRH1ADRA1B
SCHEMBL8042425 0.79 DRD2 (0.63) DRD2ADRA1AHRH1ADRA1B
SCHEMBL4429177 0.75 UTS2R (0.57) DRD2HTR2AMCHR1CHRM1KCNH2
SCHEMBL8013233 0.75 CHRM1 (0.61) DRD2HTR2AMCHR1CHRM1KCNH2
SCHEMBL8045751 0.75 DRD2 (0.61) DRD2CHRM1CHRM2CHRM4CHRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6133275-A ALPHA 1 ADRENORECEPTOR ANTAGONISTS; TREATING BENIGN PROSTATIC HYPERPLASIA AND OTHER UROLOGICAL DISEASES E.G., BLADDER OUTLET OBSTRUCTION), NEUROGENIC BLADDER AND GYNECOLOGICAL SYNDROMES, E.G., DYSMENORRHEA; UTERINE MUSCLE RELAXANTS ABBOTT LABORATORIES (US) 2000-10-17 US disclosed
WO-1999057122-A1 3-PHENYLPYRROLE ALPHA-1 ADRENERGIC COMPOUNDS ABBOTT LABORATORIES (US) 1999-11-11 WO disclosed