SCHEMBL8042494

SCHEMBL8042494

Cn1c(Sc2ncc(C(=O)O)s2)nnc1-c1cccs1

nearest known ligand 0.56

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.56
CYP3A4 P08684 1/20 0.56
KDM4E B2RXH2 2/20 0.53
NPC1 O15118 4/20 0.53
RAB9A P51151 4/20 0.53
MIF P14174 1/20 0.51
TSHR P16473 4/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
ALDH1A1 P00352 4/20 0.47
NPSR1 Q6W5P4 2/20 0.47
KMT2A Q03164 3/20 0.46
POLB P06746 2/20 0.46
MAPT P10636 2/20 0.46
GAA P10253 1/20 0.46
ALPG P10696 1/20 0.46
MEN1 O00255 2/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
USP2 O75604 1/20 0.43
HSD17B10 Q99714 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8034049 0.85 TSHR (0.58) CYP3A4KDM4ETSHRALDH1A1NPSR1
SCHEMBL8041830 0.83 CPB1 (0.47) CYP3A4KDM4ENPC1RAB9ATSHR
SCHEMBL8045746 0.83 KMT2A (0.53) HDAC6CYP3A4KDM4ENPC1RAB9A
SCHEMBL8046882 0.83 RECQL (0.41) HDAC6CYP3A4KDM4ENPC1RAB9A
SCHEMBL8042001 0.82 HSD17B10 (0.50) HDAC6CYP3A4KDM4ETSHRALDH1A1
SCHEMBL8041833 0.82 ALDH1A1 (0.46) CYP3A4KDM4ENPC1RAB9ATSHR
SCHEMBL8048062 0.81 KDM4E (0.58) HDAC6CYP3A4KDM4ENPC1RAB9A
SCHEMBL8050851 0.81 TSHR (0.49) HDAC6CYP3A4KDM4ETSHRALDH1A1
SCHEMBL8050243 0.81 NPSR1 (0.57) CYP3A4KDM4ETSHRALDH1A1NPSR1
SCHEMBL8043876 0.81 RECQL (0.50) CYP3A4KDM4ENPC1RAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed