SCHEMBL8043296

SCHEMBL8043296

O=[N+]([O-])c1cnc(Sc2nnc(SCc3cccc(C(F)(F)F)c3)s2)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATG4B Q9Y4P1 1/20 0.50
MAPK8 P45983 8/20 0.48
MAPK9 P45984 8/20 0.48
MAPK10 P53779 1/20 0.48
ALDH1A1 P00352 4/20 0.46
LMNA P02545 3/20 0.46
HTT P42858 3/20 0.46
POLB P06746 1/20 0.46
MAPT P10636 3/20 0.45
NR1D1 P20393 1/20 0.43
NR1H3 Q13133 1/20 0.43
RAB9A P51151 2/20 0.41
DAO P14920 1/20 0.41
NPC1 O15118 1/20 0.40
S1PR4 O95977 1/20 0.40
HSP90AA1 P07900 1/20 0.40
S1PR1 P21453 1/20 0.40
MAPK1 P28482 1/20 0.40
AGTR1 P30556 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8043300 0.77 MAPK8 (0.47) ATG4BMAPK8MAPK9MAPK10ALDH1A1
SCHEMBL11430427 0.75 MAPK8 (0.79) MAPK8MAPK9MAPK10ALDH1A1LMNA
SCHEMBL8037040 0.73 MAPK8 (0.67) ATG4BMAPK8MAPK9MAPK10ALDH1A1
SCHEMBL8046264 0.73 MAPK8 (0.64) ATG4BMAPK8MAPK9MAPK10ALDH1A1
SCHEMBL3909244 0.72 NPC1 (0.50) ALDH1A1LMNAHTTRAB9ANPC1
SCHEMBL6097608 0.72 RAB9A (0.50) ALDH1A1LMNAHTTMAPTRAB9A
SCHEMBL8044444 0.71 ALDH1A1 (0.44) ATG4BMAPK8MAPK9MAPK10ALDH1A1
SCHEMBL8050694 0.71 MAPK8 (0.61) ATG4BMAPK8MAPK9MAPK10ALDH1A1
SCHEMBL8032483 0.71 MAPK8 (0.57) ATG4BMAPK8MAPK9MAPK10ALDH1A1
SCHEMBL8042714 0.70 MAPK8 (0.60) MAPK8MAPK9MAPK10ALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143765-A ENZYME IHIBITORS OF PROTEIN SUGEN, INC. (US) 2000-11-07 US disclosed
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed