SCHEMBL8044444

SCHEMBL8044444

O=[N+]([O-])c1cnc(Sc2nnnn2-c2cccc(C(F)(F)F)c2)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.44
MAPT P10636 5/20 0.44
HTT P42858 4/20 0.44
GAA P10253 1/20 0.44
PKM P14618 1/20 0.44
ATG4B Q9Y4P1 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.40
USP2 O75604 1/20 0.40
LMNA P02545 1/20 0.40
ALPG P10696 1/20 0.40
MAPK8 P45983 2/20 0.40
MAPK9 P45984 2/20 0.40
MAPK10 P53779 2/20 0.40
KEAP1 Q14145 1/20 0.40
NFE2L2 Q16236 1/20 0.40
NPSR1 Q6W5P4 3/20 0.39
NPC1 O15118 3/20 0.39
RAB9A P51151 3/20 0.39
TLR9 Q9NR96 3/20 0.39
MAPK1 P28482 3/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8032753 0.85 SMN1; SMN2 (0.51) ALDH1A1MAPTHTTGAAPKM
SCHEMBL8046704 0.84 ALDH1A1 (0.60) ALDH1A1MAPTHTTGAAPKM
SCHEMBL8048205 0.83 ALDH1A1 (0.42) ALDH1A1MAPTHTTGAASMN1; SMN2
SCHEMBL8046515 0.81 POLB (0.45) ALDH1A1MAPTHTTGAASMN1; SMN2
SCHEMBL8045713 0.81 ALDH1A1 (0.48) ALDH1A1MAPTHTTGAAPKM
SCHEMBL8046724 0.80 ALDH1A1 (0.40) ALDH1A1MAPTHTTSMN1; SMN2LMNA
SCHEMBL8034759 0.80 MAPT (0.47) ALDH1A1MAPTHTTGAAPKM
SCHEMBL8032487 0.80 ALDH1A1 (0.44) ALDH1A1MAPTHTTGAAPKM
SCHEMBL8178174 0.80 MAPK8 (0.62) ALDH1A1MAPTHTTGAAATG4B
SCHEMBL8041923 0.79 PDK1 (0.47) ALDH1A1MAPTHTTGAAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed
WO-1998027092-A1 THIAZOLE COMPOUNDS AND METHODS OF MODULATING SIGNAL TRANSDUCTION SUGEN, INC. (US) 1998-06-25 WO disclosed