SCHEMBL8043794

SCHEMBL8043794

Cc1ncccc1-c1c[c]ccn1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
TDO2 P48775 1/20 0.39
VHL P40337 1/20 0.34
PDPK1 O15530 1/20 0.34
PDE2A O00408 2/20 0.33
PDE10A Q9Y233 2/20 0.33
DHODH Q02127 1/20 0.33
ELANE P08246 1/20 0.33
PDE4D Q08499 1/20 0.33
PDE3A Q14432 1/20 0.33
BLM P54132 2/20 0.32
KDM4E B2RXH2 1/20 0.32
LMNA P02545 1/20 0.32
CYP1A2 P05177 1/20 0.32
POLB P06746 1/20 0.32
CCR1 P32246 1/20 0.32
CCR5 P51681 1/20 0.32
CCR8 P51685 1/20 0.32
METAP1 P53582 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7162849 0.77 BTK (0.44) PDE2APDE10ADHODHELANEKDM4E
SCHEMBL2752958 0.76 NUDT1 (0.39) MKNK2PDPK1P2RX7GAANPC1
SCHEMBL1450105 0.76 MKNK1 (0.45) MKNK1MKNK2TDO2VHLPDE2A
SCHEMBL5148218 0.76 KDM4E (0.54) MKNK1MKNK2TDO2VHLPDE10A
SCHEMBL31469002 0.75 MKNK1 (0.52) MKNK1MKNK2TDO2VHLPDE2A
SCHEMBL3421959 0.75 MKNK1 (0.52) MKNK1MKNK2TDO2VHLPDE2A
SCHEMBL2156047 0.73 MKNK1 (0.53) MKNK1MKNK2TDO2VHLPDE2A
SCHEMBL2751007 0.73 CDK2 (0.38) PDE10ANPC1
SCHEMBL1450328 0.72 KDM4E (0.36) BLMKDM4ELMNACYP1A2POLB
SCHEMBL4976600 0.72 ALDH1A1 (0.44) BLMKDM4ELMNACYP1A2POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6107301-A PSYCHOLOGICAL DISORDERS DUPONT PHARMACEUTICALS COMPANY (US) 2000-08-22 US disclosed