SCHEMBL8044240

SCHEMBL8044240

CC(C)(C)c1nc(Sc2nnnn2-c2ccc([N+](=O)[O-])s2)sc1Br

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.35
SMN1; SMN2 Q16637 5/20 0.33
LMNA P02545 4/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
ALDH1A1 P00352 8/20 0.33
MITF O75030 2/20 0.33
RECQL P46063 1/20 0.33
MAPT P10636 5/20 0.32
PSMD14 O00487 1/20 0.32
HTT P42858 3/20 0.32
GAA P10253 1/20 0.32
PKM P14618 1/20 0.32
MAPK1 P28482 2/20 0.31
MEN1 O00255 2/20 0.31
USP2 O75604 1/20 0.31
ALPG P10696 1/20 0.31
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8049792 0.86 KMT2A (0.35) KMT2ASMN1; SMN2LMNACYP1A2CYP3A4
SCHEMBL8050561 0.84 ALDH1A1 (0.34) KMT2ASMN1; SMN2LMNAALDH1A1MAPT
SCHEMBL8041914 0.83 ALDH1A1 (0.33) KMT2ASMN1; SMN2LMNAALDH1A1MAPT
SCHEMBL8042693 0.78 ALDH1A1 (0.35) KMT2ASMN1; SMN2LMNAALDH1A1MAPT
SCHEMBL8047853 0.78 KMT2A (0.40) KMT2ASMN1; SMN2LMNACYP1A2CYP3A4
SCHEMBL8034587 0.78 RECQL (0.37) KMT2ASMN1; SMN2LMNACYP1A2CYP3A4
SCHEMBL8042628 0.76 ALDH1A1 (0.41) KMT2ASMN1; SMN2LMNAALDH1A1RECQL
SCHEMBL8043561 0.76 ALDH1A1 (0.52) KMT2ASMN1; SMN2LMNAALDH1A1MAPT
SCHEMBL8043929 0.76 MAPK8 (0.47) KMT2ASMN1; SMN2LMNAALDH1A1MAPT
SCHEMBL8042232 0.76 ALDH1A1 (0.50) KMT2ASMN1; SMN2LMNACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed