SCHEMBL8044571

SCHEMBL8044571

COc1nsc(NC(=O)N[C@@H](CC(C)C)C(=O)NC(=O)CC(C)C)n1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 7/20 0.41
MMP3 P08254 1/20 0.40
LMNA P02545 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
TP53 P04637 1/20 0.38
MAPT P10636 1/20 0.38
MAPK1 P28482 1/20 0.38
RAB9A P51151 1/20 0.38
MEN1 O00255 1/20 0.37
STAT3 P40763 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7455524 0.84 ALDH1A1 (0.46) ANPEPMMP3LMNAALDH1A1TP53
SCHEMBL8044575 0.83 CAPN1 (0.41) ANPEPMMP3LMNAMAPK1
SCHEMBL7642642 0.77 ALDH1A1 (0.40) LMNASMN1; SMN2NPC1ALDH1A1TP53
SCHEMBL7406417 0.74 ALDH1A1 (0.37) LMNASMN1; SMN2NPC1ALDH1A1TP53
Proline SCHEMBL7402744 0.72 ALDH1A1 (0.36) MMP3LMNAALDH1A1MAPTMAPK1
SCHEMBL7442154 0.71 CYP2C9 (0.43)
SCHEMBL7402896 0.71 ALDH1A1 (0.36) MMP3LMNAALDH1A1MAPTMAPK1
Proline SCHEMBL7402894 0.71 SMN1; SMN2 (0.39) MMP3SMN1; SMN2
SCHEMBL7397791 0.70 SMN1; SMN2 (0.34) LMNASMN1; SMN2NPC1ALDH1A1TP53
SCHEMBL22436168 0.68 ADORA3 (0.40) SMN1; SMN2NPC1TP53MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114537-A 1,2,4-THIADIAZOLE COMPOUND IS USEFUL FOR TRAPPING THIOL COMPOUNDS AND SELECTIVELY CHANGING THIOLS TO DISULFIDE COMPOUNDS APOTEX INC. (CA) 2000-09-05 US disclosed