SCHEMBL8044639

SCHEMBL8044639

Cn1c(Sc2nc(C(F)(F)F)c(C(=O)O)s2)nnc1-c1cccs1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 2/20 0.49
CYP3A4 P08684 1/20 0.49
NPC1 O15118 5/20 0.48
RAB9A P51151 5/20 0.48
KDM4E B2RXH2 2/20 0.48
MIF P14174 1/20 0.47
ALDH1A1 P00352 5/20 0.43
POLB P06746 3/20 0.43
NPSR1 Q6W5P4 2/20 0.43
TSHR P16473 4/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
KMT2A Q03164 2/20 0.43
MAPT P10636 2/20 0.43
GAA P10253 1/20 0.43
ALPG P10696 1/20 0.43
HSD17B10 Q99714 2/20 0.42
USP2 O75604 1/20 0.42
MEN1 O00255 1/20 0.42
ALOX15 P16050 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8047063 0.86 TSHR (0.51) CYP3A4KDM4EALDH1A1NPSR1TSHR
SCHEMBL8042695 0.85 CPB1 (0.43) CYP3A4NPC1RAB9AKDM4EALDH1A1
SCHEMBL8042411 0.85 KMT2A (0.39) CYP3A4NPC1RAB9AKDM4EMIF
SCHEMBL8051659 0.85 KMT2A (0.49) HDAC6CYP3A4NPC1RAB9AKDM4E
SCHEMBL8042697 0.84 ALDH1A1 (0.43) CYP3A4NPC1RAB9AKDM4EALDH1A1
SCHEMBL8050842 0.84 HSD17B10 (0.46) CYP3A4KDM4EALDH1A1POLBNPSR1
SCHEMBL8047548 0.84 NPSR1 (0.54) CYP3A4KDM4EALDH1A1NPSR1TSHR
SCHEMBL8042509 0.83 HSD17B10 (0.47) CYP3A4KDM4EALDH1A1POLBNPSR1
SCHEMBL8047020 0.83 RECQL (0.47) CYP3A4NPC1RAB9AKDM4EALDH1A1
SCHEMBL8047418 0.83 KMT2A (0.38) HDAC6CYP3A4NPC1RAB9AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed