SCHEMBL8042695

SCHEMBL8042695

O=C(O)c1sc(Sc2nnc(-c3cccs3)n2CCc2ccccc2)nc1C(F)(F)F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CPB1 P15086 1/20 0.43
USP2 O75604 2/20 0.43
HPGD P15428 1/20 0.43
RAB9A P51151 4/20 0.42
NPC1 O15118 3/20 0.41
TSHR P16473 4/20 0.40
LMNA P02545 3/20 0.40
HTT P42858 2/20 0.40
ALDH1A1 P00352 5/20 0.40
MAPT P10636 4/20 0.40
SMN1; SMN2 Q16637 3/20 0.40
POLB P06746 2/20 0.40
HSD17B10 Q99714 2/20 0.40
GALR3 O60755 1/20 0.40
ESR2 Q92731 1/20 0.40
CTDSP1 Q9GZU7 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GAA P10253 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP3A4 P08684 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8051659 0.85 KMT2A (0.49) HPGDRAB9ANPC1TSHRHTT
SCHEMBL8042411 0.85 KMT2A (0.39) CPB1HPGDRAB9ANPC1TSHR
SCHEMBL8044639 0.85 HDAC6 (0.49) USP2RAB9ANPC1TSHRALDH1A1
SCHEMBL8047063 0.83 TSHR (0.51) USP2HPGDTSHRHTTALDH1A1
SCHEMBL8047418 0.83 KMT2A (0.38) CPB1HPGDRAB9ANPC1TSHR
SCHEMBL8042697 0.81 ALDH1A1 (0.43) HPGDRAB9ANPC1TSHRLMNA
SCHEMBL8033984 0.79 RAB9A (0.45) CPB1USP2HPGDRAB9ANPC1
SCHEMBL8041830 0.79 CPB1 (0.47) CPB1USP2HPGDRAB9ANPC1
SCHEMBL8042509 0.79 HSD17B10 (0.47) USP2HPGDTSHRHTTALDH1A1
SCHEMBL8044326 0.78 NPSR1 (0.47) USP2HPGDTSHRHTTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed