SCHEMBL8044749

SCHEMBL8044749

O=[N+]([O-])c1cc2c(c(Cl)c1OCc1ccccc1)CCCC2

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIN1 Q13526 2/20 0.44
POLB P06746 1/20 0.42
PTGES O14684 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ATM Q13315 1/20 0.38
MAOB P27338 3/20 0.38
MAOA P21397 2/20 0.38
MAPT P10636 2/20 0.37
MGMT P16455 1/20 0.37
TDP1 Q9NUW8 1/20 0.37
CTSV O60911 1/20 0.36
CTSL P07711 1/20 0.36
RXRA P19793 2/20 0.36
RXRB P28702 2/20 0.36
RXRG P48443 2/20 0.36
CYP19A1 P11511 1/20 0.36
AR P10275 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL629645 0.86 POLB (0.42) PIN1POLBPTGESMEN1KMT2A
SCHEMBL27921821 0.83 POLB (0.42) PIN1POLBPTGESMEN1KMT2A
SCHEMBL8044819 0.79 TSHR (0.40) RAB9AMAOBMAOAMAPTTDP1
SCHEMBL8031159 0.78 PIN1 (0.48) PIN1POLBMEN1KMT2ANPC1
SCHEMBL629877 0.75 POLB (0.55) PIN1POLBMEN1KMT2ANPC1
SCHEMBL27940470 0.74 DHODH (0.44) POLBMAOBMAOAMAPTMGMT
SCHEMBL6178097 0.71 PIN1 (0.49) PIN1POLBPTGESMEN1KMT2A
SCHEMBL27388637 0.70 HTR1A (0.55) PIN1POLBMEN1KMT2ANPC1
SCHEMBL4928212 0.70 MAPT (0.55) PIN1POLBMEN1KMT2ANPC1
SCHEMBL8041772 0.70 HPGD (0.39) POLBMEN1KMT2ANPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686144-B1 NEW COMPOUNDS UNIV MARYLAND (US) 2000-04-19 EP disclosed
US-5688945-A Compounds ASTRA AKTIEBOLAG (SE) 1997-11-18 US disclosed
US-5661183-A 3-hydroxy anthanilic acid derivatives THE UNIVERSITY OF MARYLAND (US) 1997-08-26 US disclosed
EP-0686144-A1 NEW COMPOUNDS Astra Aktiebolag (SE) 1995-12-13 EP disclosed
WO-1994019315-A1 NEW COMPOUNDS ASTRA AKTIEBOLAG (SE) 1994-09-01 WO disclosed