SCHEMBL8041772

SCHEMBL8041772

O=C(/C=N/O)Nc1cc2c(c(Cl)c1OCc1ccccc1)CCCC2

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.39
MAPK1 P28482 1/20 0.39
DHODH Q02127 1/20 0.39
NPC1 O15118 2/20 0.39
RAB9A P51151 2/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
CYP1A2 P05177 1/20 0.37
NPSR1 Q6W5P4 1/20 0.37
NLRP3 Q96P20 2/20 0.36
RXRB P28702 5/20 0.36
RXRA P19793 4/20 0.36
RXRG P48443 4/20 0.36
LMNA P02545 1/20 0.36
ACHE P22303 4/20 0.36
KDM4E B2RXH2 1/20 0.35
POLB P06746 1/20 0.35
NFKB1 P19838 1/20 0.35
NFKB2 Q00653 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8031094 0.81 MAPK1 (0.47) HPGDMAPK1NPC1RAB9ASMN1; SMN2
SCHEMBL8044819 0.72 TSHR (0.40) DHODHRAB9ASMN1; SMN2RXRBRXRA
SCHEMBL8044749 0.70 PIN1 (0.44) NPC1RAB9AMEN1KMT2ARXRB
SCHEMBL4829038 0.68 ALDH1A1 (0.56) HPGDSMN1; SMN2MEN1KMT2ALMNA
SCHEMBL12359714 0.68 ALDH1A1 (0.56) HPGDSMN1; SMN2MEN1KMT2ALMNA
SCHEMBL2479933 0.66 ALDH1A1 (0.52) HPGDMEN1KMT2ACYP1A2NPSR1
SCHEMBL31417705 0.66 ALDH1A1 (0.52) HPGDMEN1KMT2ACYP1A2NPSR1
SCHEMBL2251499 0.66 ALDH1A1 (0.52) HPGDMEN1KMT2ACYP1A2NPSR1
SCHEMBL11888126 0.66 ALDH1A1 (0.52) HPGDMEN1KMT2ACYP1A2NPSR1
SCHEMBL8043075 0.65 DHODH (0.43) HPGDDHODHRXRBRXRARXRG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0686144-B1 NEW COMPOUNDS UNIV MARYLAND (US) 2000-04-19 EP disclosed
US-5688945-A Compounds ASTRA AKTIEBOLAG (SE) 1997-11-18 US disclosed
US-5661183-A 3-hydroxy anthanilic acid derivatives THE UNIVERSITY OF MARYLAND (US) 1997-08-26 US disclosed
EP-0686144-A1 NEW COMPOUNDS Astra Aktiebolag (SE) 1995-12-13 EP disclosed
WO-1994019315-A1 NEW COMPOUNDS ASTRA AKTIEBOLAG (SE) 1994-09-01 WO disclosed