SCHEMBL8044783

SCHEMBL8044783

O=C(Cc1ccc(O)cc1)c1ccc(Br)cc1

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.68
RAB9A P51151 4/20 0.68
GAA P10253 3/20 0.60
MAPT P10636 2/20 0.60
LMNA P02545 1/20 0.60
ALOX12 P18054 1/20 0.60
HSP90AA1 P07900 1/20 0.54
KCNH2 Q12809 1/20 0.54
GSK3B P49841 2/20 0.53
PTPN1 P18031 1/20 0.53
CA2 P00918 2/20 0.50
ALOX15 P16050 1/20 0.50
HDAC3 O15379 1/20 0.50
HDAC4 P56524 1/20 0.50
HDAC1 Q13547 1/20 0.50
HDAC7 Q8WUI4 1/20 0.50
HDAC2 Q92769 1/20 0.50
HDAC10 Q969S8 1/20 0.50
HDAC11 Q96DB2 1/20 0.50
HDAC8 Q9BY41 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7854876 1.00 NPC1 (0.68) NPC1RAB9AGAAMAPTLMNA
SCHEMBL29985867 0.92 GSK3B (0.61) NPC1RAB9AGAAMAPTLMNA
SCHEMBL8584136 0.92 GSK3B (0.61) NPC1RAB9AGAAMAPTLMNA
SCHEMBL1642242 0.90 NPC1 (0.81) NPC1RAB9AGAAMAPTLMNA
SCHEMBL12835116 0.84 RAB9A (0.72) NPC1RAB9AGAAMAPTLMNA
SCHEMBL5318356 0.83 RAB9A (0.71) NPC1RAB9AMAPTLMNAGSK3B
SCHEMBL13959588 0.83 ALDH1A1 (0.52) NPC1RAB9AGAAMAPTLMNA
SCHEMBL6199282 0.83 PTPN1 (0.55) NPC1RAB9AGAAMAPTLMNA
SCHEMBL6201625 0.83 RAB9A (0.71) NPC1RAB9AMAPTLMNAGSK3B
SCHEMBL6203410 0.83 PTPN1 (0.55) NPC1RAB9AGAAMAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0636367-B1 Use of phenylalkylamines for producing cholesterol lowering agents HOFFMANN LA ROCHE (CH) 2000-03-29 EP disclosed
US-5637771-A Compound useful for lowering cholesterol HOFFMANN-LA ROCHE INC. (US) 1997-06-10 US disclosed
US-5574071-A ADMINISTERING PHENYLALKYLAMINO KETONES HOFFMANN-LA ROCHE INC. (US) 1996-11-12 US disclosed
US-5495048-A ANTICHOLESTEROL AGENTS HOFFMANN-LA ROCHE INC. (US) 1996-02-27 US disclosed
EP-0636367-A1 Use of phenylalkylamines for producing cholesterol lowering agents F. HOFFMANN-LA ROCHE AG (CH) 1995-02-01 EP disclosed