SCHEMBL8044926

SCHEMBL8044926

O=C(c1ccc(Cl)cc1)C(O)[C@H]1O[C@@H](Cl)C[C@@]1(O)C(=O)c1ccc(Cl)cc1

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.32
PTGS2 P35354 1/20 0.32
GSK3B P49841 1/20 0.31
CES2 O00748 1/20 0.31
CES1 P23141 1/20 0.31
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30
SLC6A3 Q01959 1/20 0.30
ALOX15 P16050 1/20 0.30
TSHR P16473 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9594501 1.00 P2RX7 (0.32) P2RX7PTGS2GSK3BCES2CES1
SCHEMBL11350296 1.00 P2RX7 (0.32) P2RX7PTGS2GSK3BCES2CES1
SCHEMBL16446965 0.89 HPGD (0.33) CES2CES1MEN1GAAKMT2A
SCHEMBL9614440 0.89 HPGD (0.33) CES2CES1MEN1GAAKMT2A
SCHEMBL11104413 0.89 HPGD (0.33) CES2CES1MEN1GAAKMT2A
SCHEMBL3268947 0.84 P2RX7 (0.30) P2RX7PTGS2
SCHEMBL5971739 0.83 HPGD (0.34) P2RX7PTGS2SLC6A3
SCHEMBL1799676 0.82 TDP1 (0.33)
SCHEMBL2476289 0.78 GSK3B (0.32) P2RX7GSK3BCES2CES1MEN1
SCHEMBL2476284 0.78 GSK3B (0.32) P2RX7GSK3BCES2CES1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0635517-B1 Process for Producing 1-(2'-deoxy-beta-D-erythropentofuranosyl)-5-trifluoromethyluracil Derivatives MITSUI CHEMICALS INC (JP) 2000-05-17 EP disclosed
EP-0990651-A1 Process for producing 5-trifluoromethyluracil derivatives Mitsui Chemicals, Inc. (JP) 2000-04-05 EP disclosed
US-5532349-A ANTITUMOR, VIRICIDES MITSUI TOATSU CHEMICALS, INC. (JP) 1996-07-02 US disclosed
EP-0635517-A1 Process for Producing 1-(2'-deoxy-beta-D-erythropentofuranosyl)-5-trifluoromethyluracil Derivatives MITSUI TOATSU CHEMICALS, Inc. (JP) 1995-01-25 EP disclosed