SCHEMBL8045133

SCHEMBL8045133

[c]1nccc(Sc2ccccc2)n1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 3/20 0.39
HTT P42858 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.35
PLK4 O00444 2/20 0.33
ALDH1A1 P00352 6/20 0.33
PTGIR P43119 1/20 0.33
MAPT P10636 3/20 0.32
SMN1; SMN2 Q16637 3/20 0.32
MGLL Q99685 1/20 0.32
HSD17B10 Q99714 1/20 0.32
NPSR1 Q6W5P4 3/20 0.32
LMNA P02545 2/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
GRM5 P41594 1/20 0.32
NOTUM Q6P988 1/20 0.32
NCOA1 Q15788 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9414589 0.84 DDAH1 (0.50) ALDH1A1MAPTLMNAMEN1KMT2A
SCHEMBL558374 0.70
SCHEMBL6543651 0.69 HPGD (0.40) HPGDHTTL3MBTL1ALDH1A1MAPT
SCHEMBL30634505 0.66 L3MBTL1 (0.70) HPGDHTTL3MBTL1ALDH1A1MAPT
SCHEMBL2225278 0.66 L3MBTL1 (0.70) HPGDHTTL3MBTL1ALDH1A1MAPT
SCHEMBL9216740 0.65 DDAH1 (0.41) HPGDHTTALDH1A1PTGIRMAPT
SCHEMBL8569111 0.65
SCHEMBL3284927 0.65 HTT (0.44) HPGDHTTL3MBTL1PLK4ALDH1A1
SCHEMBL8429277 0.64 HPGD (0.52) HPGDHTTL3MBTL1PLK4ALDH1A1
Diphenylsulfane SCHEMBL11466727 0.64 HPGD (0.53) HPGDHTTALDH1A1PTGIRMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6100268-A MIGRAINES JANSSEN PHARMACEUTICA, N.V. (BE) 2000-08-08 US disclosed
US-5824682-A Vasoconstrictive dihydrobenzopyran derivatives JANSSEN PHARMACEUTICA, N.V. (BE) 1998-10-20 US disclosed
EP-0714396-A1 VASOCONTRICTIVE DIHYDROBENZOPYRAN DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1996-06-05 EP disclosed
WO-1995005383-A1 VASOCONTRICTIVE DIHYDROBENZOPYRAN DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1995-02-23 WO disclosed