SCHEMBL8045157

SCHEMBL8045157

CCc1cc2c(cc1C(=O)OC)NC(C)(C)S2(=O)=O

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 13/20 0.34
KDM4E B2RXH2 11/20 0.34
LMNA P02545 5/20 0.34
MAPT P10636 7/20 0.33
HSD17B10 Q99714 5/20 0.33
HPGD P15428 5/20 0.33
GAA P10253 3/20 0.33
HTT P42858 2/20 0.33
TSHR P16473 2/20 0.33
ALOX15 P16050 1/20 0.33
GLA P06280 2/20 0.32
CASP1 P29466 1/20 0.31
CASP7 P55210 1/20 0.31
ATM Q13315 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
KMT2A Q03164 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8056504 0.75 IRAK4 (0.35) ALDH1A1KDM4ELMNAMAPTHSD17B10
SCHEMBL8062949 0.74 ALDH1A1 (0.34) ALDH1A1KDM4ELMNAMAPTHSD17B10
SCHEMBL8056970 0.73 ALDH1A1 (0.33) ALDH1A1KDM4ELMNAMAPTHSD17B10
SCHEMBL8056980 0.70 TSHR (0.34) ALDH1A1KDM4ELMNAMAPTHSD17B10
SCHEMBL8056991 0.70 ALDH1A1 (0.33) ALDH1A1KDM4ELMNAMAPTHSD17B10
SCHEMBL8057086 0.69 ALDH1A1 (0.32) ALDH1A1KDM4ELMNAMAPTHSD17B10
SCHEMBL8060805 0.68 RXRA (0.33) ALDH1A1KDM4ELMNAMAPTHSD17B10
SCHEMBL8060722 0.68 ALDH1A1 (0.36) ALDH1A1KDM4ELMNAMAPTHSD17B10
SCHEMBL8062745 0.68 ALDH1A1 (0.34) ALDH1A1KDM4ELMNAMAPTHSD17B10
SCHEMBL8062814 0.68 ALDH1A1 (0.35) ALDH1A1KDM4ELMNAMAPTHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed