SCHEMBL8062814

SCHEMBL8062814

CCc1cc2c(cc1C(=O)OC)S(=O)(=O)C(C)(C)CO2

nearest known ligand 0.50

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.35
KDM4E B2RXH2 10/20 0.35
KMT2A Q03164 5/20 0.35
MEN1 O00255 3/20 0.35
TSHR P16473 2/20 0.35
RAB9A P51151 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
RARB P10826 1/20 0.34
RARG P13631 1/20 0.34
NPC1 O15118 1/20 0.34
MAPT P10636 3/20 0.33
HSD17B10 Q99714 3/20 0.33
HTT P42858 1/20 0.33
HPGD P15428 4/20 0.33
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
LMNA P02545 2/20 0.32
TP53 P04637 1/20 0.31
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8058204 0.85 ALDH1A1 (0.37) ALDH1A1KDM4EKMT2AMEN1TSHR
SCHEMBL8056991 0.81 ALDH1A1 (0.33) ALDH1A1KDM4EKMT2ATSHRMAPT
SCHEMBL8060815 0.79 KDM4E (0.38) ALDH1A1KDM4EKMT2AMEN1TSHR
SCHEMBL8056980 0.78 TSHR (0.34) ALDH1A1KDM4EKMT2ATSHRMAPT
SCHEMBL8056280 0.77 KDM4E (0.43) ALDH1A1KDM4EKMT2AMEN1TSHR
SCHEMBL8056352 0.76 RARB (0.46) ALDH1A1KDM4EKMT2AMEN1TSHR
SCHEMBL8060805 0.76 RXRA (0.33) ALDH1A1KDM4EKMT2AMEN1TSHR
SCHEMBL8060881 0.75 ALDH1A1 (0.35) ALDH1A1KDM4EKMT2AMEN1TSHR
SCHEMBL8057340 0.75 TSHR (0.34) ALDH1A1KDM4ETSHRRARBRARG
SCHEMBL8045260 0.75 ALDH1A1 (0.33) ALDH1A1KDM4EKMT2AMEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed