SCHEMBL8045258

SCHEMBL8045258

CCc1cc2c(cc1C(=O)OC)S(=O)(=O)CC21OCCO1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 1/20 0.33
PDGFRA P16234 1/20 0.33
ACVR1B P36896 1/20 0.33
PIK3CA P42336 1/20 0.33
RIPK1 Q13546 1/20 0.33
RIPK3 Q9Y572 1/20 0.33
ALDH1A1 P00352 7/20 0.33
KDM4E B2RXH2 6/20 0.33
HSD17B10 Q99714 4/20 0.33
HTT P42858 1/20 0.33
MAPT P10636 1/20 0.33
KMT2A Q03164 2/20 0.32
REV1 Q9UBZ9 1/20 0.32
MEN1 O00255 1/20 0.32
TSHR P16473 2/20 0.32
HPGD P15428 2/20 0.32
LMNA P02545 2/20 0.32
HCRTR1 O43613 1/20 0.32
HCRTR2 O43614 1/20 0.32
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8062769 0.85 PDGFRA (0.34) BRAFPDGFRAACVR1BPIK3CARIPK1
SCHEMBL8062997 0.84 PIK3CA (0.34) BRAFPDGFRAACVR1BPIK3CARIPK1
SCHEMBL8062746 0.82 RXRA (0.36) ALDH1A1KDM4EHSD17B10HTTMAPT
SCHEMBL8062776 0.81 ALDH1A1 (0.34) ALDH1A1KDM4EHSD17B10HTTMAPT
SCHEMBL8045064 0.81 CFTR (0.36) BRAFPDGFRAACVR1BPIK3CARIPK1
SCHEMBL8060847 0.80
SCHEMBL8062982 0.80 ALDH1A1 (0.34) ALDH1A1KDM4EHSD17B10HTTMAPT
SCHEMBL8057402 0.79 ALDH1A1 (0.36) ALDH1A1KDM4EHSD17B10HTTMAPT
SCHEMBL8062745 0.79 ALDH1A1 (0.34) ALDH1A1KDM4EHSD17B10HTTMAPT
SCHEMBL8056978 0.79 RXRA (0.34) ALDH1A1KDM4EHSD17B10HTTMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed