SCHEMBL8062997

SCHEMBL8062997

COC(=O)c1cc2c(cc1F)C1(CS2(=O)=O)OCCO1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 2/20 0.34
BRAF P15056 1/20 0.34
PDGFRA P16234 1/20 0.34
ACVR1B P36896 1/20 0.34
RIPK1 Q13546 1/20 0.34
RIPK3 Q9Y572 1/20 0.34
PKM P14618 2/20 0.33
PIK3CD O00329 1/20 0.33
AKT1 P31749 1/20 0.33
PIK3CB P42338 1/20 0.33
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 4/20 0.33
WDR5 P61964 1/20 0.31
GAA P10253 1/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
GLA P06280 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8062769 0.86 PDGFRA (0.34) PIK3CABRAFPDGFRAACVR1BRIPK1
SCHEMBL8045064 0.84 CFTR (0.36) PIK3CABRAFPDGFRAACVR1BRIPK1
SCHEMBL8045258 0.84 BRAF (0.33) PIK3CABRAFPDGFRAACVR1BRIPK1
SCHEMBL8045039 0.82 RARB (0.35) ALDH1A1KDM4EGAAHPGDTSHR
SCHEMBL8045253 0.78 ALDH1A1 (0.43) ALDH1A1KDM4EGAAHPGDTSHR
SCHEMBL21032580 0.73 PKM (0.34) PKMALDH1A1KDM4EWDR5GAA
SCHEMBL522786 0.71 CA12 (0.47) ALDH1A1KDM4EGAAHPGDTSHR
SCHEMBL410165 0.67 ALPL (0.45) PKMALDH1A1KDM4EGAAHPGD
SCHEMBL8058193 0.67 VEGFA (0.41) PKMALDH1A1KDM4EGAAHPGD
SCHEMBL8058138 0.67 KDM4E (0.36) PDGFRAALDH1A1KDM4EGAAHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6028069-A Heterocyclyl-condensed benzoylguanidines, their production and use as inhibitors of the cellular Na+/H+-antiporter MERCK PATENT GESELLSCHAFT MIT BERSCHRANKER HAFTUNG (DE) 2000-02-22 US disclosed