SCHEMBL8045552

SCHEMBL8045552

NC1=NC(c2cccn2Cc2ccccc2)Cc2ccsc21

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 13/20 0.58
NOS3 P29474 10/20 0.58
ACHE P22303 4/20 0.36
HTR1A P08908 3/20 0.36
HTR6 P50406 3/20 0.36
HTR7 P34969 2/20 0.36
BCHE P06276 3/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8098153 0.99 NOS2 (0.57) NOS2NOS3ACHEHTR1AHTR6
Hydrochloric Acid SCHEMBL8090054 0.73 NOS3 (0.97) NOS2NOS3
Hydrochloric Acid SCHEMBL8106647 0.67 NOS2 (0.97) NOS2NOS3
SCHEMBL8057607 0.65 NOS2 (1.00) NOS2NOS3
SCHEMBL8057623 0.65 NOS2 (0.56) NOS2NOS3
Hydrochloric Acid SCHEMBL8100105 0.64 NOS2 (0.97) NOS2NOS3
SCHEMBL8045503 0.64 NOS2 (1.00) NOS2NOS3
Hydrochloric Acid SCHEMBL8107228 0.64 NOS2 (0.55) NOS2NOS3
Hydrochloric Acid SCHEMBL8099873 0.64 NOS2 (0.97) NOS2NOS3
SCHEMBL8233735 0.64 NOS2 (0.71) NOS2NOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1027052-A1 NOVEL COMBINATION AstraZeneca UK Limited (GB) 2000-08-16 EP claimed
US-6046191-A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF AND AN AMIDINE COMPOUND; FOR TREATMENT OF INFLAMMATORY DISORDERS ASTRA PHARMACEUTICALS LTD. (GB) 2000-04-04 US claimed
WO-1999018960-A1 NOVEL COMBINATION ASTRAZENECA UK LIMITED (GB) 1999-04-22 WO claimed
EP-1027052-A1 NOVEL COMBINATION AstraZeneca UK Limited (GB) 2000-08-16 EP disclosed
US-6046191-A PHARMACEUTICAL COMBINATION COMPRISING A COX-2 INHIBITOR OR A PHARMACEUTICALLY ACCEPTABLE SALT THEREOF AND AN AMIDINE COMPOUND; FOR TREATMENT OF INFLAMMATORY DISORDERS ASTRA PHARMACEUTICALS LTD. (GB) 2000-04-04 US disclosed
WO-1999018960-A1 NOVEL COMBINATION ASTRAZENECA UK LIMITED (GB) 1999-04-22 WO disclosed