SCHEMBL8046007

SCHEMBL8046007

CCSC1=C(C(=O)O)N2C(=O)[C@H]([C@@H](C)O[Si](C)(C)C(C)(C)C)[C@H]2[C@H]1C

nearest known ligand 0.42

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
CACNA1C Q13936 1/20 0.36
FAP Q12884 1/20 0.33
ESR1 P03372 1/20 0.33
PTGS1 P23219 1/20 0.33
PDE4A P27815 1/20 0.33
ELANE P08246 4/20 0.31
KDM4E B2RXH2 1/20 0.30
LMNA P02545 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428941 0.88 CACNA1C (0.36) CACNA1CFAPESR1PTGS1PDE4A
SCHEMBL9427855 0.88 CACNA1C (0.36) CACNA1CFAPESR1PTGS1PDE4A
SCHEMBL9428111 0.86 ELANE (0.36) CACNA1CESR1PTGS1PDE4AELANE
SCHEMBL8839225 0.84 ELANE (0.31) CACNA1CELANE
SCHEMBL30006016 0.84 ELANE (0.31) CACNA1CELANE
SCHEMBL8038860 0.83 ESR1 (0.37) CACNA1CFAPESR1PTGS1PDE4A
SCHEMBL9834843 0.83 ESR1 (0.37) CACNA1CFAPESR1PTGS1PDE4A
SCHEMBL9698199 0.82 ELANE (0.31) CACNA1CELANE
SCHEMBL8046011 0.81 MAPT (0.35) KDM4ELMNA
SCHEMBL8975911 0.81 MAPT (0.35) KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0587436-B1 Process for preparing carbapenem and penem compounds and new compounds involved in that process SANKYO CO (JP) 2000-05-10 EP disclosed
US-5614624-A THIO SUBSTITUTED, ANTIBIOTICS, CHEMICAL INTERMEDIATES SANKYO COMPANY, LIMITED (JP) 1997-03-25 US disclosed
US-5541317-A PENICILLIN DERIVATIVES, CYCLIZATION OF ESTERS OR THIOESTERS SANKYO COMPANY, LIMITED (JP) 1996-07-30 US disclosed
EP-0587436-A1 Process for preparing carbapenem and penem compounds and new compounds involved in that process SANKYO COMPANY LIMITED (JP) 1994-03-16 EP disclosed