SCHEMBL8046642

SCHEMBL8046642

CC(C)(C)c1nc(Sc2nnc(C(C)(C)C)n2-c2ccccc2)sc1Br

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.36
KMT2A Q03164 3/20 0.36
HTT P42858 3/20 0.36
MEN1 O00255 2/20 0.36
MAPT P10636 2/20 0.36
RAB9A P51151 1/20 0.36
TSHR P16473 2/20 0.34
SMN1; SMN2 Q16637 3/20 0.32
NPSR1 Q6W5P4 1/20 0.32
USP2 O75604 1/20 0.32
TP53 P04637 2/20 0.31
KDM4E B2RXH2 2/20 0.31
HSD17B10 Q99714 2/20 0.31
SLC22A12 Q96S37 2/20 0.31
VCP P55072 3/20 0.30
RXRA P19793 1/20 0.30
RXRB P28702 1/20 0.30
RXRG P48443 1/20 0.30
LMNA P02545 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050859 0.89 ALDH1A1 (0.35) ALDH1A1KMT2AHTTMEN1MAPT
SCHEMBL8043099 0.82 TSHR (0.57) ALDH1A1KMT2AHTTMEN1MAPT
SCHEMBL8043571 0.82 ATM (0.43) ALDH1A1KMT2AHTTMEN1TSHR
SCHEMBL8716255 0.81 TP53 (0.43) ALDH1A1KMT2AHTTMEN1RAB9A
SCHEMBL8042649 0.80 ALDH1A1 (0.36) ALDH1A1KMT2AHTTMEN1MAPT
SCHEMBL8044131 0.80 RPA1 (0.44) ALDH1A1KMT2AHTTMEN1MAPT
SCHEMBL8050718 0.80 HTT (0.51) ALDH1A1KMT2AHTTMEN1MAPT
SCHEMBL8043752 0.79 KDM4E (0.48) ALDH1A1KMT2AHTTMEN1MAPT
SCHEMBL8043561 0.79 ALDH1A1 (0.52) ALDH1A1KMT2AHTTMAPTRAB9A
SCHEMBL8044820 0.78

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed