SCHEMBL8043752

SCHEMBL8043752

Cc1nc(-c2ccccc2)sc1-c1nnc(Sc2nc(C(C)(C)C)c(Br)s2)n1-c1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 10/20 0.48
ALDH1A1 P00352 9/20 0.48
CYP2C9 P11712 4/20 0.48
HPGD P15428 3/20 0.48
CYP1A2 P05177 2/20 0.48
RAB9A P51151 4/20 0.46
SMN1; SMN2 Q16637 4/20 0.46
MAPT P10636 2/20 0.46
CYP2C19 P33261 2/20 0.43
CYP3A4 P08684 2/20 0.43
CYP2D6 P10635 1/20 0.43
LMNA P02545 3/20 0.37
APOBEC3G Q9HC16 1/20 0.37
NPC1 O15118 3/20 0.36
TSHR P16473 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
COMT P21964 1/20 0.35
HDAC6 Q9UBN7 1/20 0.35
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8050065 0.88 KDM4E (0.52) KDM4EALDH1A1CYP2C9HPGDCYP1A2
SCHEMBL8042708 0.80 ALDH1A1 (0.52) KDM4EALDH1A1CYP2C9HPGDCYP1A2
SCHEMBL8047964 0.80 KDM4E (0.54) KDM4EALDH1A1CYP2C9HPGDCYP1A2
SCHEMBL8044969 0.80 ALDH1A1 (0.45) KDM4EALDH1A1CYP2C9HPGDCYP1A2
SCHEMBL8043099 0.79 TSHR (0.57) KDM4EALDH1A1CYP2C9HPGDCYP1A2
SCHEMBL8043571 0.79 ATM (0.43) ALDH1A1HPGDSMN1; SMN2TSHRMEN1
SCHEMBL8046642 0.79 ALDH1A1 (0.36) KDM4EALDH1A1RAB9ASMN1; SMN2MAPT
SCHEMBL8034048 0.79 KDM4E (0.53) KDM4EALDH1A1CYP2C9HPGDCYP1A2
SCHEMBL8716255 0.78 TP53 (0.43) KDM4EALDH1A1HPGDCYP1A2RAB9A
SCHEMBL8044821 0.78 ALDH1A1 (0.47) KDM4EALDH1A1CYP2C9HPGDCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed