SCHEMBL8046975

SCHEMBL8046975

c1ccc(-n2c(Cc3c[nH]c4ccccc34)nnc2Sc2nccs2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GPR84 Q9NQS5 7/20 0.43
BACE1 P56817 1/20 0.42
MET P08581 3/20 0.40
SSTR1 P30872 2/20 0.40
SSTR4 P31391 2/20 0.40
SSTR3 P32745 2/20 0.40
GLA P06280 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
GHSR Q92847 1/20 0.39
CYP3A4 P08684 1/20 0.39
MAPT P10636 1/20 0.39
AHR P35869 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8045394 0.83 GPR84 (0.48) GPR84BACE1METSSTR1SSTR4
SCHEMBL8033967 0.83 CYP1A2 (0.42) GPR84BACE1SSTR1SSTR4SSTR3
SCHEMBL8050059 0.82 GPR84 (0.43) GPR84BACE1METSSTR1SSTR4
SCHEMBL8033920 0.81 HTT (0.49) GPR84BACE1SSTR1SSTR4SSTR3
SCHEMBL8034186 0.80 MET (0.41) GPR84BACE1METSSTR1SSTR4
SCHEMBL8043560 0.80 BACE1 (0.45) GPR84BACE1METSSTR1SSTR4
SCHEMBL8049951 0.79 GPR84 (0.42) GPR84BACE1METSSTR1SSTR4
SCHEMBL8051882 0.79 BACE1 (0.44) GPR84BACE1GHSRALDH1A1CYP1A2
SCHEMBL8045236 0.79 SSTR4 (0.41) GPR84BACE1METSSTR1SSTR4
SCHEMBL8042613 0.79 GPR84 (0.40) GPR84BACE1METSSTR1SSTR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed