SCHEMBL8033920

SCHEMBL8033920

c1ccc(-n2c(Cc3c[nH]c4ccccc34)nnc2Sc2nc3ccccc3s2)cc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.49
ALDH1A1 P00352 3/20 0.49
NPSR1 Q6W5P4 2/20 0.49
HPGD P15428 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.48
TSHR P16473 2/20 0.44
LMNA P02545 1/20 0.44
MAPK1 P28482 1/20 0.44
GPR84 Q9NQS5 4/20 0.41
BACE1 P56817 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
SSTR1 P30872 1/20 0.40
SSTR4 P31391 1/20 0.40
SSTR3 P32745 1/20 0.40
USP2 O75604 1/20 0.39
MAPT P10636 2/20 0.39
CYP1A2 P05177 2/20 0.39
CYP2D6 P10635 2/20 0.39
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8043584 0.88 GPR84 (0.44) HTTALDH1A1NPSR1HPGDSMN1; SMN2
SCHEMBL8050073 0.87 GPR84 (0.41) HTTALDH1A1NPSR1HPGDSMN1; SMN2
SCHEMBL8050043 0.86 MAPT (0.43) HTTALDH1A1NPSR1HPGDSMN1; SMN2
SCHEMBL8041875 0.86 GPR84 (0.45) HTTALDH1A1NPSR1HPGDSMN1; SMN2
SCHEMBL8034186 0.85 MET (0.41) ALDH1A1GPR84BACE1SSTR1SSTR4
SCHEMBL8033967 0.82 CYP1A2 (0.42) ALDH1A1GPR84BACE1SSTR1SSTR4
SCHEMBL8045394 0.82 GPR84 (0.48) ALDH1A1GPR84BACE1SSTR1SSTR4
SCHEMBL8046381 0.82 GHSR (0.39) ALDH1A1LMNAGPR84BACE1SSTR1
SCHEMBL8050059 0.82 GPR84 (0.43) ALDH1A1GPR84BACE1SSTR1SSTR4
SCHEMBL8046975 0.81 GPR84 (0.43) ALDH1A1SMN1; SMN2GPR84BACE1SSTR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed