SCHEMBL8048253

SCHEMBL8048253

CCCc1nnc(Sc2nc3ccccc3s2)s1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.52
MAPT P10636 4/20 0.52
LMNA P02545 3/20 0.52
FBP1 P09467 2/20 0.51
CYP1A2 P05177 4/20 0.49
CYP2D6 P10635 3/20 0.49
MAPK1 P28482 3/20 0.49
CYP2C19 P33261 3/20 0.49
CYP3A4 P08684 2/20 0.49
HIF1A Q16665 1/20 0.49
L3MBTL1 Q9Y468 1/20 0.49
HSD17B10 Q99714 5/20 0.49
HPGD P15428 3/20 0.49
ADRA2A P08913 1/20 0.49
ADORA3 P0DMS8 1/20 0.49
DRD2 P14416 1/20 0.49
ALOX15 P16050 1/20 0.49
ADRA2B P18089 1/20 0.49
ADRA2C P18825 1/20 0.49
DRD1 P21728 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8043241 0.93 FBP1 (0.50) ALDH1A1MAPTLMNAFBP1CYP1A2
SCHEMBL8046503 0.89 HSD17B10 (0.55) ALDH1A1MAPTLMNAFBP1CYP1A2
SCHEMBL8044052 0.86 MAPK1 (0.49) ALDH1A1MAPTLMNAFBP1CYP1A2
SCHEMBL8033602 0.85 CYP1A2 (0.48) ALDH1A1MAPTLMNAFBP1CYP1A2
SCHEMBL8044035 0.83 HSD17B10 (0.51) ALDH1A1MAPTLMNAFBP1CYP1A2
SCHEMBL8049883 0.82 CYP1A2 (0.48) ALDH1A1MAPTLMNAFBP1CYP1A2
SCHEMBL8043628 0.82 HPGD (0.59) ALDH1A1MAPTFBP1CYP1A2CYP2D6
SCHEMBL8043621 0.81 GLA (0.51) ALDH1A1MAPTLMNAMAPK1L3MBTL1
SCHEMBL8042757 0.81 CYP1A2 (0.53) ALDH1A1MAPTLMNAFBP1CYP1A2
SCHEMBL8045797 0.79 HSP90AA1 (0.45) ALDH1A1MAPTLMNAMAPK1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed