SCHEMBL8049883

SCHEMBL8049883

COCc1nnc(Sc2nc3ccccc3s2)s1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 5/20 0.48
CYP2C19 P33261 4/20 0.48
CYP2D6 P10635 3/20 0.48
CYP3A4 P08684 3/20 0.48
MAPK1 P28482 2/20 0.48
L3MBTL1 Q9Y468 2/20 0.48
HIF1A Q16665 1/20 0.48
ALDH1A1 P00352 6/20 0.47
HSD17B10 Q99714 4/20 0.47
HPGD P15428 4/20 0.47
FBP1 P09467 2/20 0.47
ADRA2A P08913 1/20 0.47
ADORA3 P0DMS8 1/20 0.47
DRD2 P14416 1/20 0.47
ALOX15 P16050 1/20 0.47
ADRA2B P18089 1/20 0.47
ADRA2C P18825 1/20 0.47
DRD1 P21728 1/20 0.47
MC5R P33032 1/20 0.47
OPRM1 P35372 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8046503 0.85 HSD17B10 (0.55) CYP1A2CYP2C19CYP2D6CYP3A4MAPK1
SCHEMBL8048253 0.82 ALDH1A1 (0.52) CYP1A2CYP2C19CYP2D6CYP3A4MAPK1
SCHEMBL8044035 0.82 HSD17B10 (0.51) CYP1A2CYP2C19CYP2D6CYP3A4MAPK1
SCHEMBL8043241 0.81 FBP1 (0.50) CYP1A2CYP2C19CYP2D6CYP3A4MAPK1
SCHEMBL8032726 0.80 LMNA (0.40) MAPK1ALDH1A1HSD17B10HPGDTDP1
SCHEMBL8042757 0.80 CYP1A2 (0.53) CYP1A2CYP2C19CYP2D6CYP3A4MAPK1
SCHEMBL8044052 0.80 MAPK1 (0.49) CYP1A2CYP2C19CYP2D6CYP3A4MAPK1
SCHEMBL8050213 0.78 PKM (0.44) ALDH1A1HSD17B10HPGDSMN1; SMN2LMNA
SCHEMBL8045054 0.78 LMNA (0.43) ALDH1A1HSD17B10HPGDTDP1SMN1; SMN2
SCHEMBL8033602 0.78 CYP1A2 (0.48) CYP1A2CYP2C19CYP2D6CYP3A4MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6080772-A 2-AMINOTHIAZOLE TRIAZOLE OR TETRAZOLE COMPOUND FOR REGULATING PROTEIN TYROSINE PHOSPHATASE ACTIVITY SUGEN, INC. (US) 2000-06-27 US disclosed